3M9Y
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![BU of 3m9y by Molmil](/molmil-images/mine/3m9y) | Crystal structure of Triosephosphate isomerase from methicillin resistant Staphylococcus aureus at 1.9 Angstrom resolution | 分子名称: | CITRIC ACID, SODIUM ION, Triosephosphate isomerase | 著者 | Mukherjee, S, Dutta, D, Saha, B, Das, A.K. | 登録日 | 2010-03-23 | 公開日 | 2011-04-06 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Crystal structures of triosephosphate isomerase from methicillin resistant Staphylococcus aureus MRSA252 provide structural insights into novel modes of ligand binding and unique conformations of catalytic loop Biochimie, 94, 2012
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2QPQ
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7PUF
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![BU of 7puf by Molmil](/molmil-images/mine/7puf) | urate oxidase azaxanthine complex under 600 bar (60 MPa) of argon | 分子名称: | 8-AZAXANTHINE, ARGON, SODIUM ION, ... | 著者 | Prange, T, Colloc'h, N, Carpentier, P. | 登録日 | 2021-09-29 | 公開日 | 2022-02-09 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.86 Å) | 主引用文献 | Comparative study of the effects of high hydrostatic pressure per se and high argon pressure on urate oxidase ligand stabilization Acta Cryst. D, 78, 2022
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6GC9
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6GCA
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6GCC
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![BU of 6gcc by Molmil](/molmil-images/mine/6gcc) | Crystal structure of glutathione transferase Xi 3 mutant C56S from Trametes versicolor in complex with dextran-sulfate | 分子名称: | 3,4-di-O-sulfo-alpha-D-glucopyranose-(1-6)-3,4-di-O-sulfo-alpha-D-altropyranose-(1-6)-1,2,3,4-tetra-O-sulfo-alpha-D-allopyranose, Glutathione transferase Xi 3 mutant C56S | 著者 | Schwartz, M, Favier, F, Didierjean, C. | 登録日 | 2018-04-17 | 公開日 | 2018-08-29 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Trametes versicolor glutathione transferase Xi 3, a dual Cys-GST with catalytic specificities of both Xi and Omega classes. FEBS Lett., 592, 2018
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6HTA
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![BU of 6hta by Molmil](/molmil-images/mine/6hta) | Crystal structure of glutathione transferase Xi 3 mutant C56S from Trametes versicolor | 分子名称: | ACETATE ION, DIMETHYL SULFOXIDE, Glutathione transferase Xi 3 C56S | 著者 | Schwartz, M, Favier, F, Didierjean, C. | 登録日 | 2018-10-03 | 公開日 | 2018-10-10 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Trametes versicolor glutathione transferase Xi 3, a dual Cys-GST with catalytic specificities of both Xi and Omega classes. FEBS Lett., 592, 2018
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4H35
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3IMX
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![BU of 3imx by Molmil](/molmil-images/mine/3imx) | Crystal Structure of human glucokinase in complex with a synthetic activator | 分子名称: | (2R)-3-cyclopentyl-N-(5-methoxy[1,3]thiazolo[5,4-b]pyridin-2-yl)-2-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}propanamide, Glucokinase, SODIUM ION, ... | 著者 | Stams, T, Vash, B. | 登録日 | 2009-08-11 | 公開日 | 2009-10-06 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Investigation of functionally liver selective glucokinase activators for the treatment of type 2 diabetes. J.Med.Chem., 52, 2009
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6GCB
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4FW8
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![BU of 4fw8 by Molmil](/molmil-images/mine/4fw8) | Crystal structure of FABG4 complexed with Coenzyme NADH | 分子名称: | (2S,5R,8R,11S,14S,17S,21R)-5,8,11,14,17-PENTAMETHYL-4,7,10,13,16,19-HEXAOXADOCOSANE-2,21-DIOL, 1,4-DIHYDRONICOTINAMIDE ADENINE DINUCLEOTIDE, 3-oxoacyl-(Acyl-carrier-protein) reductase | 著者 | Dutta, D, Bhattacharyya, S, Das, A.K. | 登録日 | 2012-06-30 | 公開日 | 2012-11-28 | 最終更新日 | 2024-03-20 | 実験手法 | X-RAY DIFFRACTION (2.79 Å) | 主引用文献 | Crystal structure of hexanoyl-CoA bound to beta-ketoacyl reductase FabG4 of Mycobacterium tuberculosis Biochem.J., 450, 2013
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4N8D
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![BU of 4n8d by Molmil](/molmil-images/mine/4n8d) | DPP4 complexed with syn-7aa | 分子名称: | 1-(cis-1-phenyl-4-{[(2E)-3-phenylprop-2-en-1-yl]oxy}cyclohexyl)methanamine, 2-acetamido-2-deoxy-beta-D-glucopyranose, Dipeptidyl peptidase 4, ... | 著者 | Ostermann, N, Zink, F, Kroemer, M. | 登録日 | 2013-10-17 | 公開日 | 2014-02-12 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | Discovery of C-(1-aryl-cyclohexyl)-methylamines as selective, orally available inhibitors of dipeptidyl peptidase IV. Bioorg.Med.Chem.Lett., 24, 2014
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4N8E
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![BU of 4n8e by Molmil](/molmil-images/mine/4n8e) | DPP4 complexed with compound 12a | 分子名称: | 1-[cis-4-(aminomethyl)-4-(3-chlorophenyl)cyclohexyl]piperidin-2-one, 2-acetamido-2-deoxy-beta-D-glucopyranose, Dipeptidyl peptidase 4, ... | 著者 | Ostermann, N, Zink, F, Kroemer, M. | 登録日 | 2013-10-17 | 公開日 | 2014-02-12 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Discovery of C-(1-aryl-cyclohexyl)-methylamines as selective, orally available inhibitors of dipeptidyl peptidase IV. Bioorg.Med.Chem.Lett., 24, 2014
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3V1U
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![BU of 3v1u by Molmil](/molmil-images/mine/3v1u) | Crystal structure of a beta-ketoacyl reductase FabG4 from Mycobacterium tuberculosis H37Rv complexed with NAD+ and Hexanoyl-CoA at 2.5 Angstrom resolution | 分子名称: | (2S,5R,8R,11S,14S,17S,21R)-5,8,11,14,17-PENTAMETHYL-4,7,10,13,16,19-HEXAOXADOCOSANE-2,21-DIOL, 3-oxoacyl-(Acyl-carrier-protein) reductase, HEXANOYL-COENZYME A, ... | 著者 | Dutta, D, Bhattacharyya, S, Das, A.K. | 登録日 | 2011-12-10 | 公開日 | 2012-11-28 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Crystal structure of hexanoyl-CoA bound to beta-ketoacyl reductase FabG4 of Mycobacterium tuberculosis Biochem.J., 450, 2013
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4P78
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![BU of 4p78 by Molmil](/molmil-images/mine/4p78) | HicA3 and HicB3 toxin-antitoxin complex | 分子名称: | GLYCEROL, HicA3 Toxin, HicB3 antitoxin | 著者 | Li de la Sierra-Gallay, I, Bibi-Triki, S, van Tilbeurgh, H, Lazar, N, Pradel, E. | 登録日 | 2014-03-26 | 公開日 | 2014-08-27 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.12 Å) | 主引用文献 | Functional and Structural Analysis of HicA3-HicB3, a Novel Toxin-Antitoxin System of Yersinia pestis. J.Bacteriol., 196, 2014
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4P7D
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![BU of 4p7d by Molmil](/molmil-images/mine/4p7d) | Antitoxin HicB3 crystal structure | 分子名称: | Antitoxin HicB3, CHLORIDE ION | 著者 | Li de la Sierra-Gallay, I, Bibi-Triki, S, van Tilbeurgh, H, Lazar, N, Pradel, E. | 登録日 | 2014-03-27 | 公開日 | 2014-08-27 | 最終更新日 | 2015-02-04 | 実験手法 | X-RAY DIFFRACTION (2.781 Å) | 主引用文献 | Functional and Structural Analysis of HicA3-HicB3, a Novel Toxin-Antitoxin System of Yersinia pestis. J.Bacteriol., 196, 2014
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4ALT
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![BU of 4alt by Molmil](/molmil-images/mine/4alt) | X-Ray photoreduction of Polysaccharide monooxygenase CBM33 | 分子名称: | CHITIN BINDING PROTEIN, COPPER (II) ION, DI(HYDROXYETHYL)ETHER | 著者 | Gudmundsson, M, Wu, M, Ishida, T, Momeni, M.H, Vaaje-Kolstad, G, Eijsink, V, Sandgren, M. | 登録日 | 2012-03-05 | 公開日 | 2013-02-27 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.49 Å) | 主引用文献 | Structural and Electronic Snapshots During the Transition from a Cu(II) to Cu(I) Metal Center of a Lytic Polysaccharide Monooxygenase by X-Ray Photo-Reduction. J.Biol.Chem., 289, 2014
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4BAG
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4ALS
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![BU of 4als by Molmil](/molmil-images/mine/4als) | X-Ray photoreduction of Polysaccharide monooxygenase CBM33 | 分子名称: | CHITIN BINDING PROTEIN, COPPER (II) ION, DI(HYDROXYETHYL)ETHER | 著者 | Gudmundsson, M, Wu, M, Ishida, T, Momeni, M.H, Vaaje-Kolstad, G, Eijsink, V, Sandgren, M. | 登録日 | 2012-03-05 | 公開日 | 2013-02-27 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.47 Å) | 主引用文献 | Structural and Electronic Snapshots During the Transition from a Cu(II) to Cu(I) Metal Center of a Lytic Polysaccharide Monooxygenase by X-Ray Photo-Reduction. J.Biol.Chem., 289, 2014
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4ALR
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![BU of 4alr by Molmil](/molmil-images/mine/4alr) | X-Ray photoreduction of Polysaccharide monooxygenase CBM33 | 分子名称: | CHITIN BINDING PROTEIN, COPPER (II) ION, DI(HYDROXYETHYL)ETHER | 著者 | Gudmundsson, M, Wu, M, Ishida, T, Momeni, M.H, Vaaje-Kolstad, G, Eijsink, V, Sandgren, M. | 登録日 | 2012-03-05 | 公開日 | 2013-02-27 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.49 Å) | 主引用文献 | Structural and Electronic Snapshots During the Transition from a Cu(II) to Cu(I) Metal Center of a Lytic Polysaccharide Monooxygenase by X-Ray Photo-Reduction. J.Biol.Chem., 289, 2014
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4ALC
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![BU of 4alc by Molmil](/molmil-images/mine/4alc) | X-Ray photoreduction of Polysaccharide monooxigenase CBM33 | 分子名称: | CHITIN BINDING PROTEIN, COPPER (II) ION, DI(HYDROXYETHYL)ETHER | 著者 | Gudmundsson, M, Wu, M, Ishida, T, Momeni, M.H, Vaaje-Kolstad, G, Eijsink, V, Sandgren, M. | 登録日 | 2012-03-02 | 公開日 | 2013-02-27 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.49 Å) | 主引用文献 | Structural and Electronic Snapshots During the Transition from a Cu(II) to Cu(I) Metal Center of a Lytic Polysaccharide Monooxygenase by X-Ray Photo-Reduction. J.Biol.Chem., 289, 2014
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4ALE
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![BU of 4ale by Molmil](/molmil-images/mine/4ale) | Structure changes of Polysaccharide monooxygenase CBM33A from Enterococcus faecalis by X-ray induced photoreduction. | 分子名称: | CHITIN BINDING PROTEIN, COPPER (II) ION, DI(HYDROXYETHYL)ETHER | 著者 | Gudmundsson, M, Wu, M, Ishida, T, Momeni, M.H, Vaaje-Kolstad, G, Eijsink, V, Sandgren, M. | 登録日 | 2012-03-02 | 公開日 | 2013-02-27 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.48 Å) | 主引用文献 | Structural and Electronic Snapshots During the Transition from a Cu(II) to Cu(I) Metal Center of a Lytic Polysaccharide Monooxygenase by X-Ray Photo-Reduction. J.Biol.Chem., 289, 2014
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4ALQ
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![BU of 4alq by Molmil](/molmil-images/mine/4alq) | X-Ray photoreduction of Polysaccharide monooxygenase CBM33 | 分子名称: | CHITIN BINDING PROTEIN, COPPER (II) ION, DI(HYDROXYETHYL)ETHER | 著者 | Gudmundsson, M, Wu, M, Ishida, T, Momeni, M.H, Vaaje-Kolstad, G, Eijsink, V, Sandgren, M. | 登録日 | 2012-03-05 | 公開日 | 2013-02-27 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.48 Å) | 主引用文献 | Structural and Electronic Snapshots During the Transition from a Cu(II) to Cu(I) Metal Center of a Lytic Polysaccharide Monooxygenase by X-Ray Photo-Reduction. J.Biol.Chem., 289, 2014
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4CW3
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![BU of 4cw3 by Molmil](/molmil-images/mine/4cw3) | Crystal structure of cofactor-free urate oxidase in complex with the 5-peroxo derivative of 9-metyl uric acid (X-ray dose, 665 kGy) | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, (5S)-5-(dioxidanyl)-9-methyl-7H-purine-2,6,8-trione, 9-METHYL URIC ACID, ... | 著者 | Bui, S, Steiner, R.A. | 登録日 | 2014-04-01 | 公開日 | 2014-10-29 | 最終更新日 | 2018-02-21 | 実験手法 | X-RAY DIFFRACTION (1.34 Å) | 主引用文献 | Direct evidence for a peroxide intermediate and a reactive enzyme-substrate-dioxygen configuration in a cofactor-free oxidase. Angew. Chem. Int. Ed. Engl., 53, 2014
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4CW6
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![BU of 4cw6 by Molmil](/molmil-images/mine/4cw6) | Crystal structure of cofactor-free urate oxidase in complex with the 5-peroxo derivative of 9-metyl uric acid (X-ray dose, 92 kGy) | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, (5S)-5-(dioxidanyl)-9-methyl-7H-purine-2,6,8-trione, 9-METHYL URIC ACID, ... | 著者 | Bui, S, Steiner, R.A. | 登録日 | 2014-04-01 | 公開日 | 2014-10-29 | 最終更新日 | 2018-02-21 | 実験手法 | X-RAY DIFFRACTION (1.28 Å) | 主引用文献 | Direct evidence for a peroxide intermediate and a reactive enzyme-substrate-dioxygen configuration in a cofactor-free oxidase. Angew. Chem. Int. Ed. Engl., 53, 2014
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