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3EAP
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BU of 3eap by Molmil
Crystal structure of the RhoGAP domain of ARHGAP11A
分子名称: Rho GTPase-activating protein 11A, UNKNOWN ATOM OR ION
著者Shen, Y, Shen, L, Tong, Y, Tempel, W, MacKenzie, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Weigelt, J, Bochkarev, A, Park, H, Structural Genomics Consortium, Structural Genomics Consortium (SGC)
登録日2008-08-26
公開日2008-09-02
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal structure of the RhoGAP domain of ARHGAP11A
To be Published
3F2R
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BU of 3f2r by Molmil
Crystal structure of human choline kinase alpha in complex with hemicholinium-3
分子名称: (2S,2'S)-2,2'-biphenyl-4,4'-diylbis(2-hydroxy-4,4-dimethylmorpholin-4-ium), Choline kinase alpha, UNKNOWN ATOM OR ION
著者Hong, B, Tempel, W, Rabeh, W.M, MacKenzie, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Weigelt, J, Bochkarev, A, Park, H, Structural Genomics Consortium (SGC)
登録日2008-10-30
公開日2008-11-11
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Crystal structure of human choline kinase alpha in complex with hemicholinium-3
To be Published
3FK2
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BU of 3fk2 by Molmil
Crystal structure of the RhoGAP domain of human glucocorticoid receptor DNA-binding factor 1
分子名称: Glucocorticoid receptor DNA-binding factor 1, UNKNOWN ATOM OR ION
著者Nedyalkova, L, Tong, Y, Tempel, W, Loppnau, P, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Weigelt, J, Bochkarev, A, Park, H, Structural Genomics Consortium (SGC)
登録日2008-12-15
公開日2008-12-23
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Crystal structure of the RhoGAP domain of human glucocorticoid receptor DNA-binding factor 1
To be Published
3FI8
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BU of 3fi8 by Molmil
Crystal structure of choline kinase from Plasmodium Falciparum, PF14_0020
分子名称: ADENOSINE-5'-DIPHOSPHATE, Choline kinase, MAGNESIUM ION, ...
著者Wernimont, A.K, Pizarro, J.C, Artz, J.D, Amaya, M.F, Xiao, T, Lew, J, Wasney, G, Senesterra, G, Kozieradzki, I, Cossar, D, Vedadi, M, Schapira, M, Bochkarev, A, Arrowsmith, C.H, Bountra, C, Weigelt, J, Edwards, A.M, Hui, R, Hills, T, Structural Genomics Consortium (SGC)
登録日2008-12-11
公開日2009-02-10
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal structure of choline kinase from Plasmodium Falciparum, PF14_0020
TO BE PUBLISHED
3F3Z
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BU of 3f3z by Molmil
Crystal structure of Cryptosporidium parvum calcium dependent protein kinase cgd7_1840 in presence of indirubin E804
分子名称: 3-({[(3S)-3,4-dihydroxybutyl]oxy}amino)-1H,2'H-2,3'-biindol-2'-one, Calcium/calmodulin-dependent protein kinase with a kinase domain and 4 calmodulin like EF hands, GLYCEROL
著者Wernimont, A.K, Lew, J, Wasney, G, Kozieradzki, I, Cossar, D, Vedadi, M, Bochkarev, A, Arrowsmith, C.H, Sundstrom, M, Weigelt, J, Edwards, A.M, Hui, R, Artz, J.D, Amani, M, Structural Genomics Consortium (SGC)
登録日2008-10-31
公開日2008-12-23
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.84 Å)
主引用文献Crystal structure of Cryptosporidium parvum calcium dependent protein kinase cgd7_1840 in presence of indirubin E804
To be Published
3FB3
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BU of 3fb3 by Molmil
Crystal Structure of Trypanosoma Brucei Acetyltransferase, Tb11.01.2886
分子名称: N-acetyltransferase
著者Wernimont, A.K, Marino, K, Zhang, A.Z, Ma, D, Lin, Y.H, MacKenzie, F, Kozieradzki, I, Cossar, D, Zhao, Y, Schapira, M, Bochkarev, A, Arrowsmith, C.H, Bountra, C, Weigelt, J, Edwards, A.M, Ferguson, M.A.J, Hui, R, Qiu, W, Structural Genomics Consortium (SGC)
登録日2008-11-18
公開日2008-11-25
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Crystal Structure of Trypanosoma Brucei Acetyltransferase, Tb11.01.2886
TO BE PUBLISHED
3EZ3
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BU of 3ez3 by Molmil
Crystal Structure of Plasmodium vivax geranylgeranylpyrophosphate synthase PVX_092040 with zoledronate and IPP bound
分子名称: 1,2-ETHANEDIOL, 3-METHYLBUT-3-ENYL TRIHYDROGEN DIPHOSPHATE, Farnesyl pyrophosphate synthase, ...
著者Wernimont, A.K, Lew, J, Zhao, Y, Kozieradzki, I, Cossar, D, Schapira, M, Bochkarev, A, Arrowsmith, C.H, Bountra, C, Weigelt, J, Edwards, A.M, Hui, R, Artz, J.D, Structural Genomics Consortium (SGC)
登録日2008-10-22
公開日2008-12-02
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.304 Å)
主引用文献Crystal Structure of Plasmodium vivax geranylgeranylpyrophosphate synthase PVX_092040 with zoledronate and IPP bound
TO BE PUBLISHED
3FL2
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BU of 3fl2 by Molmil
Crystal structure of the ring domain of the E3 ubiquitin-protein ligase UHRF1
分子名称: E3 ubiquitin-protein ligase UHRF1, ZINC ION
著者Walker, J.R, Avvakumov, G.V, Xue, S, Li, Y, Bountra, C, Weigelt, J, Arrowsmith, C.H, Edwards, A.M, Bochkarev, A, Dhe-Paganon, S, Structural Genomics Consortium (SGC)
登録日2008-12-18
公開日2009-01-20
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Structure of the Ring Domain of the E3 Ubiquitin-Protein Ligase Uhrf1
To be Published
3DL9
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BU of 3dl9 by Molmil
Crystal structure of CYP2R1 in complex with 1-alpha-hydroxy-vitamin D2
分子名称: (1S,3R,5Z,7E,22E)-9,10-secoergosta-5,7,10,22-tetraene-1,3-diol, Cycloheptakis-(1-4)-(alpha-D-glucopyranose), Cytochrome P450 2R1, ...
著者Strushkevich, N.V, Tempel, W, Gilep, A.A, Loppnau, P, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Wilkstrom, M, Bochkarev, A, Park, H, Structural Genomics Consortium (SGC)
登録日2008-06-26
公開日2008-08-05
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.721 Å)
主引用文献Crystal structure of CYP2R1 in complex with 1-alpha-hydroxy-vitamin D2.
To be Published
3DLM
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BU of 3dlm by Molmil
Crystal structure of Tudor domain of human Histone-lysine N-methyltransferase SETDB1
分子名称: Histone-lysine N-methyltransferase SETDB1
著者Amaya, M.F, Dombrovski, L, Loppnau, P, Bountra, C, Weigelt, J, Arrowsmith, C.H, Edwards, A.M, Bochkarev, A, Min, J, Wu, H, Structural Genomics Consortium (SGC)
登録日2008-06-27
公開日2008-08-12
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.77 Å)
主引用文献The crystal structure of Tudor domain of human Histone-lysine N-methyltransferase SETDB1.
To be Published
3DZQ
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BU of 3dzq by Molmil
Human EphA3 kinase domain in complex with inhibitor AWL-II-38.3
分子名称: EPH receptor A3, N-[2-methyl-5-({[3-(4-methyl-1H-imidazol-1-yl)-5-(trifluoromethyl)phenyl]carbonyl}amino)phenyl]isoxazole-5-carboxamide
著者Walker, J.R, Syeda, F, Gray, N, Mansoor, W, Mackenzie, F, Bountra, C, Weigelt, J, Arrowsmith, C.H, Edwards, A.M, Bochkarev, A, Dhe-Paganon, S, Structural Genomics Consortium (SGC)
登録日2008-07-30
公開日2008-08-26
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Kinase Domain of Human Ephrin Type-A Receptor 3 (Epha3) in Complex with ALW-II-38-3.
To be Published
3GFT
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BU of 3gft by Molmil
Human K-Ras (Q61H) in complex with a GTP analogue
分子名称: CITRIC ACID, GTPase KRas, MAGNESIUM ION, ...
著者Tong, Y, Tempel, W, Shen, L, Arrowsmith, C.H, Edwards, A.M, Sundstrom, M, Weigelt, J, Bochkarev, A, Park, H, Structural Genomics Consortium (SGC)
登録日2009-02-27
公開日2009-03-10
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.27 Å)
主引用文献Human K-Ras in complex with a GTP analogue
To be Published
3GBJ
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BU of 3gbj by Molmil
Crystal structure of the motor domain of kinesin KIF13B bound with ADP
分子名称: ADENOSINE-5'-DIPHOSPHATE, KIF13B protein, MAGNESIUM ION, ...
著者Tong, Y, Shen, L, Shen, Y, Tempel, W, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Weigelt, J, Bochkarev, A, Park, H, Structural Genomics Consortium (SGC)
登録日2009-02-19
公開日2009-03-03
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.102 Å)
主引用文献Crystal structure of the motor domain of kinesin KIF13B bound with ADP
To be Published
3DKO
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BU of 3dko by Molmil
Complex between the kinase domain of human ephrin type-a receptor 7 (epha7) and inhibitor alw-ii-49-7
分子名称: 5-[(2-methyl-5-{[3-(trifluoromethyl)phenyl]carbamoyl}phenyl)amino]pyridine-3-carboxamide, Ephrin type-A receptor 7
著者Walker, J.R, Syeda, F, Gray, N, Butler-Cole, C, Bountra, C, Wolkstrom, M, Arrowsmith, C.H, Edwards, A.M, Bochkarev, A, Dhe-Paganon, S, Structural Genomics Consortium (SGC)
登録日2008-06-25
公開日2008-08-19
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Kinase domain of human ephrin type-a receptor 7 (epha7) in complex with ALW-II-49-7
To be Published
3DWD
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BU of 3dwd by Molmil
Crystal structure of the ArfGAP domain of human ARFGAP1
分子名称: ADP-ribosylation factor GTPase-activating protein 1, UNKNOWN ATOM OR ION, ZINC ION
著者Nedyalkova, L, Tong, Y, Tempel, W, Landry, R, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Wilkstrom, M, Bochkarev, A, Park, H, Structural Genomics Consortium (SGC)
登録日2008-07-22
公開日2008-08-05
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Crystal structure of the ArfGAP domain of human ARFGAP1
To be Published
3GUC
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BU of 3guc by Molmil
Human Ubiquitin-activating Enzyme 5 in Complex with AMPPNP
分子名称: PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, Ubiquitin-like modifier-activating enzyme 5, ZINC ION
著者Walker, J.R, Bacik, J.P, Li, Y, Weigelt, J, Bountra, C, Arrowsmith, C.H, Edwards, A.M, Bochkarev, A, Dhe-Paganon, S, Structural Genomics Consortium (SGC)
登録日2009-03-29
公開日2009-05-26
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献Human Ubiquitin-activating Enzyme 5 in Complex with AMPPNP
To be Published
3H6N
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BU of 3h6n by Molmil
Crystal Structure of the ubiquitin-like domain of plexin D1
分子名称: ARSENIC, Plexin-D1, UNKNOWN ATOM OR ION
著者Tong, Y, Nedyalkova, L, Tempel, W, MacKenzie, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Weigelt, J, Bochkarev, A, Buck, M, Park, H, Structural Genomics Consortium (SGC)
登録日2009-04-23
公開日2009-05-19
最終更新日2017-11-01
実験手法X-RAY DIFFRACTION (2.004 Å)
主引用文献Crystal Structure of the ubiquitin-like domain of plexin D1
To be Published
3H8M
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BU of 3h8m by Molmil
SAM domain of human ephrin type-a receptor 7 (EPHA7)
分子名称: Ephrin type-A receptor 7
著者Walker, J.R, Yermekbayeva, L, Butler-Cole, C, Bountra, C, Weigelt, J, Arrowsmith, C.H, Edwards, A.M, Bochkarev, A, Dhe-Paganon, S, Structural Genomics Consortium (SGC)
登録日2009-04-29
公開日2009-05-26
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献SAM Domain of Human Ephrin Type-A Receptor 7 (Epha7)
To be Published
3HIL
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BU of 3hil by Molmil
SAM Domain of Human Ephrin Type-A Receptor 1 (EphA1)
分子名称: CHLORIDE ION, Ephrin type-A receptor 1, NITRATE ION
著者Walker, J.R, Yermekbayeva, L, Butler-Cole, C, Weigelt, J, Bountra, C, Arrowsmith, C.H, Edwards, A.M, Bochkarev, A, Dhe-Paganon, S, Structural Genomics Consortium (SGC)
登録日2009-05-20
公開日2009-06-09
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献SAM Domain of Human Ephrin Type-A Receptor 1 (EphA1).
To be Published
3GUE
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BU of 3gue by Molmil
Crystal Structure of UDP-glucose phosphorylase from Trypanosoma Brucei, (Tb10.389.0330)
分子名称: (2R,3S)-1,4-DIMERCAPTOBUTANE-2,3-DIOL, GLYCEROL, SULFATE ION, ...
著者Wernimont, A.K, Marino, K, Lin, Y.H, Mackenzie, F, Kozieradzki, I, Cossar, D, Zhao, Y, Schapira, M, Bochkarev, A, Arrowsmith, C.H, Bountra, C, Weigelt, J, Edwards, A.M, Ferguson, M.A.J, Hui, R, Amani, M, Structural Genomics Consortium (SGC)
登録日2009-03-29
公開日2009-08-18
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.92 Å)
主引用文献Crystal Structure of UDP-glucose phosphorylase from Trypanosoma Brucei, (Tb10.389.0330)
To be Published
3HZJ
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BU of 3hzj by Molmil
Crystal structure of the RabGAP domain of the RABGAP1L protein
分子名称: RAB GTPase-activating protein 1-like, UNKNOWN ATOM OR ION
著者Nedyalkova, L, Tempel, W, Tong, Y, Zhong, N, MacKenzie, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Weigelt, J, Bochkarev, A, Park, H, Structural Genomics Consortium (SGC)
登録日2009-06-23
公開日2009-07-14
最終更新日2017-11-01
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal structure of the RabGAP domain of the RABGAP1L protein
To be Published
3HM5
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BU of 3hm5 by Molmil
SANT domain of human DNA methyltransferase 1 associated protein 1
分子名称: CALCIUM ION, DNA methyltransferase 1-associated protein 1, UNKNOWN ATOM OR ION
著者Dombrovski, L, Tempel, W, Amaya, M.F, Tong, Y, Ni, S, Bountra, C, Weigelt, J, Arrowsmith, C.H, Edwards, A.M, Bochkarev, A, Min, J, Park, H, Wu, H, Structural Genomics Consortium (SGC)
登録日2009-05-28
公開日2009-06-16
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献SANT domain of human DNA methyltransferase 1 associated protein 1
To be Published
3I3C
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BU of 3i3c by Molmil
Crystal Structural of CBX5 Chromo Shadow Domain
分子名称: Chromobox protein homolog 5, SODIUM ION
著者Amaya, M.F, Li, Z, Li, Y, Kozieradzki, I, Edwards, A.M, Arrowsmith, C.H, Weigelt, J, Bountra, C, Bochkarev, A, Min, J, Ouyang, H, Structural Genomics Consortium (SGC)
登録日2009-06-30
公開日2009-08-18
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.48 Å)
主引用文献Crystal Structural of CBX5 Chromo Shadow Domain
To be Published
2OWA
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BU of 2owa by Molmil
Crystal structure of putative GTPase activating protein for ADP ribosylation factor from Cryptosporidium parvum (cgd5_1040)
分子名称: Arfgap-like finger domain containing protein, ZINC ION
著者Dong, A, Lew, J, Zhao, Y, Hassanali, A, Lin, L, Ravichandran, M, Wasney, G, Vedadi, M, Kozieradzki, I, Bochkarev, A, Edwards, A.M, Arrowsmith, C.H, Weigelt, J, Sundstrom, M, Hui, R, Qiu, W, Structural Genomics Consortium (SGC)
登録日2007-02-15
公開日2007-02-27
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal structure of putative GTPase activating protein for ADP ribosylation factor from Cryptosporidium parvum (cgd5_1040)
To be Published
2ONU
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BU of 2onu by Molmil
Plasmodium falciparum ubiquitin conjugating enzyme PF10_0330, putative homologue of human UBE2H
分子名称: TETRAETHYLENE GLYCOL, Ubiquitin-conjugating enzyme, putative
著者Dong, A, Lew, J, Lin, L, Hassanali, A, Zhao, Y, Senisterra, G, Wasney, G, Vedadi, M, Kozieradzki, I, Bochkarev, A, Arrowsmith, C.H, Edwards, A.M, Sundstrom, M, Weigelt, J, Hui, R, Brokx, S.J, Structural Genomics Consortium (SGC)
登録日2007-01-24
公開日2007-02-06
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.38 Å)
主引用文献Plasmodium falciparum ubiquitin conjugating enzyme PF10_0330, putative homologue of human UBE2H
To be Published

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