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4O2A
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BU of 4o2a by Molmil
Tubulin-BAL27862 complex
Descriptor: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 3-[(4-{1-[2-(4-aminophenyl)-2-oxoethyl]-1H-benzimidazol-2-yl}-1,2,5-oxadiazol-3-yl)amino]propanenitrile, ADENOSINE-5'-DIPHOSPHATE, ...
Authors:Prota, A.E, Franck, D, Bachmann, F, Bargsten, K, Buey, R.M, Pohlmann, J, Reinelt, S, Lane, H, Steinmetz, M.O.
Deposit date:2013-12-17
Release date:2014-03-05
Last modified:2023-09-20
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:The Novel Microtubule-Destabilizing Drug BAL27862 Binds to the Colchicine Site of Tubulin with Distinct Effects on Microtubule Organization.
J.Mol.Biol., 426, 2014
4O2B
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BU of 4o2b by Molmil
Tubulin-Colchicine complex
Descriptor: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, CALCIUM ION, DI(HYDROXYETHYL)ETHER, ...
Authors:Prota, A.E, Franck, D, Bachmann, F, Bargsten, K, Buey, R.M, Pohlmann, J, Reinelt, S, Lane, H, Steinmetz, M.O.
Deposit date:2013-12-17
Release date:2014-03-05
Last modified:2023-09-20
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:The Novel Microtubule-Destabilizing Drug BAL27862 Binds to the Colchicine Site of Tubulin with Distinct Effects on Microtubule Organization.
J.Mol.Biol., 426, 2014
4AFG
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BU of 4afg by Molmil
Capitella teleta AChBP in complex with varenicline
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CAPITELLA TELETA ACHBP, VARENICLINE, ...
Authors:Brams, M, Ulens, C, Spurny, R.
Deposit date:2012-01-19
Release date:2012-05-30
Last modified:2023-12-20
Method:X-RAY DIFFRACTION (2.001 Å)
Cite:Molecular Actions of Smoking Cessation Drugs at Alpha4Beta2 Nicotinic Receptors Defined in Crystal Structures of a Homologous Binding Protein.
Proc.Natl.Acad.Sci.USA, 109, 2012
4AFH
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BU of 4afh by Molmil
Capitella teleta AChBP in complex with lobeline
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ACHBP, Alpha-Lobeline, ...
Authors:Brams, M, Ulens, C, Spurny, R.
Deposit date:2012-01-19
Release date:2012-05-30
Last modified:2023-12-20
Method:X-RAY DIFFRACTION (1.88 Å)
Cite:Molecular Actions of Smoking Cessation Drugs at Alpha4Beta2 Nicotinic Receptors Defined in Crystal Structures of a Homologous Binding Protein.
Proc.Natl.Acad.Sci.USA, 109, 2012

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