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1EAS
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BU of 1eas by Molmil
NONPEPTIDIC INHIBITORS OF HUMAN LEUKOCYTE ELASTASE. 3. DESIGN, SYNTHESIS, X-RAY CRYSTALLOGRAPHIC ANALYSIS, AND STRUCTURE-ACTIVITY RELATIONSHIPS FOR A SERIES OF ORALLY ACTIVE 3-AMINO-6-PHENYLPYRIDIN-2-ONE TRIFLUOROMETHYL KETONES
Descriptor: 3-[[(METHYLAMINO)SULFONYL]AMINO]-2-OXO-6-PHENYL-N-[3,3,3-TRIFLUORO-1-(1-METHYLETHYL)-2-OXOPHENYL]-1(2H)-PYRIDINE ACETAMIDE, PORCINE PANCREATIC ELASTASE, SODIUM ION, ...
Authors:Ceccarelli, C.
Deposit date:1994-11-22
Release date:1995-02-07
Last modified:2024-06-05
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:Nonpeptidic inhibitors of human leukocyte elastase. 3. Design, synthesis, X-ray crystallographic analysis, and structure-activity relationships for a series of orally active 3-amino-6-phenylpyridin-2-one trifluoromethyl ketones.
J.Med.Chem., 37, 1994
1EAT
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BU of 1eat by Molmil
NONPEPTIDIC INHIBITORS OF HUMAN LEUKOCYTE ELASTASE. 5. DESIGN, SYNTHESIS, AND X-RAY CRYSTALLOGRAPHY OF A SERIES OF ORALLY ACTIVE 5-AMINO-PYRIMIDIN-6-ONE-CONTAINING TRIFLUOROMETHYLKETONES
Descriptor: 2-[5-METHANESULFONYLAMINO-2-(4-AMINOPHENYL)-6-OXO-1,6-DIHYDRO-1-PYRIMIDINYL]-N-(3,3,3-TRIFLUORO-1-ISOPROPYL-2-OXOPROPYL)ACETAMIDE, PORCINE PANCREATIC ELASTASE, SODIUM ION, ...
Authors:Ceccarelli, C.
Deposit date:1994-11-22
Release date:1995-02-07
Last modified:2024-06-05
Method:X-RAY DIFFRACTION (2 Å)
Cite:Nonpeptidic inhibitors of human leukocyte elastase. 5. Design, synthesis, and X-ray crystallography of a series of orally active 5-aminopyrimidin-6-one-containing trifluoromethyl ketones.
J.Med.Chem., 38, 1995
3SQE
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BU of 3sqe by Molmil
Crystal structure of prethrombin-2 mutant S195A in the alternative form
Descriptor: GLYCEROL, Thrombin light chain, heavy chain
Authors:Pozzi, N, Chen, Z, Di Cera, E.
Deposit date:2011-07-05
Release date:2011-11-30
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:Crystal structures of prethrombin-2 reveal alternative conformations under identical solution conditions and the mechanism of zymogen activation.
Biochemistry, 50, 2011
3SQH
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BU of 3sqh by Molmil
Crystal structure of prethrombin-2 mutant S195A in the the open form
Descriptor: Thrombin light chain, heavy chain
Authors:Pozzi, N, Chen, Z, Di Cera, E.
Deposit date:2011-07-05
Release date:2011-11-30
Last modified:2023-09-13
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:Crystal structures of prethrombin-2 reveal alternative conformations under identical solution conditions and the mechanism of zymogen activation.
Biochemistry, 50, 2011
1INC
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BU of 1inc by Molmil
CRYSTAL STRUCTURES OF THE COMPLEX OF PORCINE PANCREATIC ELASTASE WITH TWO VALINE-DERIVED BENZOXAZINONE INHIBITORS
Descriptor: CALCIUM ION, PORCINE PANCREATIC ELASTASE, SULFATE ION, ...
Authors:Meyer, E.
Deposit date:1993-03-19
Release date:1994-01-31
Last modified:2024-06-05
Method:X-RAY DIFFRACTION (1.94 Å)
Cite:Crystal structures of the complex of porcine pancreatic elastase with two valine-derived benzoxazinone inhibitors.
J.Mol.Biol., 198, 1987
1JIM
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BU of 1jim by Molmil
STEREOSPECIFIC REACTION OF 3-METHOXY-4-CHLORO-7-AMINOISOCOUMARIN WITH CRYSTALLINE PORCINE PANCREATIC ELASTASE
Descriptor: METHYL(2-ACETOXY-2-(2-CARBOXY-4-AMINO-PHENYL))ACETATE, PORCINE PANCREATIC ELASTASE, SULFATE ION
Authors:Meyer, E.
Deposit date:1993-03-19
Release date:1994-01-31
Last modified:2024-06-05
Method:X-RAY DIFFRACTION (2.31 Å)
Cite:Stereospecific Reaction of 3-Methoxy-4-Chloro-7-Aminoisocoumarin with Crystalline Porcine Pancreatic Elastase
J.Am.Chem.Soc., 107, 1985
1HXF
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BU of 1hxf by Molmil
HUMAN THROMBIN COMPLEX WITH HIRUDIN VARIANT
Descriptor: HIRUDIN VARIANT, THROMBIN
Authors:Tulinsky, A, Zhang, E.
Deposit date:1996-09-09
Release date:1997-01-27
Last modified:2024-06-05
Method:X-RAY DIFFRACTION (2.1 Å)
Cite:The molecular environment of the Na+ binding site of thrombin.
Biophys.Chem., 63, 1997
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