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Estrogen Receptor Alpha Ligand Binding Domain in Complex with the Selective Estrogen Receptor Modulator Clomiphene
Descriptor:	Clomifene, Estrogen receptor
Authors:	Fanning, S.W, Greene, G.L.
Deposit date:	2020-02-03
Release date:	2020-09-16
Last modified:	2023-10-11
Method:	X-RAY DIFFRACTION (1.6 Å)
Cite:	Stereospecific lasofoxifene derivatives reveal the interplay between estrogen receptor alpha stability and antagonistic activity in ESR1 mutant breast cancer cells. Elife, 11, 2022

Bazedoxifene in Complex with Y537S Estrogen Receptor Alpha Ligand Binding Domain
Descriptor:	Bazedoxifene, Estrogen receptor
Authors:	Fanning, S.W, Greene, G.L.
Deposit date:	2019-07-12
Release date:	2019-11-20
Last modified:	2023-10-11
Method:	X-RAY DIFFRACTION (1.8 Å)
Cite:	Stereospecific lasofoxifene derivatives reveal the interplay between estrogen receptor alpha stability and antagonistic activity in ESR1 mutant breast cancer cells. Elife, 11, 2022

Estrogen Receptor Alpha Ligand Binding Domain in Complex with Raloxifene
Descriptor:	Estrogen receptor, RALOXIFENE
Authors:	Fanning, S.W.
Deposit date:	2020-10-02
Release date:	2020-11-18
Last modified:	2023-10-18
Method:	X-RAY DIFFRACTION (1.834 Å)
Cite:	Stereospecific lasofoxifene derivatives reveal the interplay between estrogen receptor alpha stability and antagonistic activity in ESR1 mutant breast cancer cells. Elife, 11, 2022