4LWH
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![BU of 4lwh by Molmil](/molmil-images/mine/4lwh) | Crystal Structure of the human Hsp90-alpha N-domain bound to the hsp90 inhibitor FJ5 | Descriptor: | Heat shock protein HSP 90-alpha, N-{3-[2,4-dihydroxy-5-(propan-2-yl)phenyl]-4-[4-(morpholin-4-ylmethyl)phenyl]-1,2-oxazol-5-yl}cyclopropanecarboxamide | Authors: | Li, J, Shi, F, Xiong, B, He, J. | Deposit date: | 2013-07-27 | Release date: | 2014-07-30 | Last modified: | 2023-11-08 | Method: | X-RAY DIFFRACTION (1.7 Å) | Cite: | Discovery of potent N-(isoxazol-5-yl)amides as HSP90 inhibitors. Eur.J.Med.Chem., 87, 2014
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3OJW
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![BU of 3ojw by Molmil](/molmil-images/mine/3ojw) | Disulfide crosslinked cytochrome P450 reductase inactive | Descriptor: | FLAVIN MONONUCLEOTIDE, FLAVIN-ADENINE DINUCLEOTIDE, NADPH-cytochrome P450 reductase | Authors: | Xia, C, Hamdane, D, Shen, A, Choi, V, Kasper, C, Zhang, H, Im, S.-C, Waskell, L, Kim, J.-J.P. | Deposit date: | 2010-08-23 | Release date: | 2011-02-23 | Last modified: | 2023-09-06 | Method: | X-RAY DIFFRACTION (2.2 Å) | Cite: | Conformational Changes of NADPH-Cytochrome P450 Oxidoreductase Are Essential for Catalysis and Cofactor Binding. J.Biol.Chem., 286, 2011
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3OJX
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![BU of 3ojx by Molmil](/molmil-images/mine/3ojx) | Disulfide crosslinked cytochrome P450 reductase inactive | Descriptor: | FLAVIN MONONUCLEOTIDE, FLAVIN-ADENINE DINUCLEOTIDE, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ... | Authors: | Xia, C, Hamdane, D, Shen, A, Choi, V, Kasper, C, Zhang, H, Im, S.-C, Waskell, L, Kim, J.-J.P. | Deposit date: | 2010-08-23 | Release date: | 2011-02-23 | Last modified: | 2023-09-06 | Method: | X-RAY DIFFRACTION (2.5 Å) | Cite: | Conformational Changes of NADPH-Cytochrome P450 Oxidoreductase Are Essential for Catalysis and Cofactor Binding. J.Biol.Chem., 286, 2011
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1Y12
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![BU of 1y12 by Molmil](/molmil-images/mine/1y12) | |
7RAG
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![BU of 7rag by Molmil](/molmil-images/mine/7rag) | |
8DP7
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![BU of 8dp7 by Molmil](/molmil-images/mine/8dp7) | |
8DP6
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![BU of 8dp6 by Molmil](/molmil-images/mine/8dp6) | |
8GYD
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![BU of 8gyd by Molmil](/molmil-images/mine/8gyd) | Structure of Schistosoma japonicum Glutathione S-transferase bound with the ligand complex of 16 | Descriptor: | (2R)-2-[[2-(5-chloranylthiophen-2-yl)-4-oxidanylidene-6-[2-(1H-1,2,3,4-tetrazol-5-yl)phenyl]quinazolin-3-yl]methyl]-3-(4-chlorophenyl)propanoic acid, ETHANOL, Glutathione S-transferase class-mu 26 kDa isozyme | Authors: | Wen, X, Jin, R, Hu, H, Zhu, J, Song, W, Lu, X. | Deposit date: | 2022-09-22 | Release date: | 2023-08-23 | Last modified: | 2023-09-13 | Method: | X-RAY DIFFRACTION (1.7 Å) | Cite: | Discovery, SAR Study of GST Inhibitors from a Novel Quinazolin-4(1 H )-one Focused DNA-Encoded Library. J.Med.Chem., 66, 2023
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4I0W
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![BU of 4i0w by Molmil](/molmil-images/mine/4i0w) | Structure of the Clostridium Perfringens CspB protease | Descriptor: | 1,2-ETHANEDIOL, CHLORIDE ION, Protease CspB, ... | Authors: | Adams, C.M, Eckenroth, B.E, Doublie, S. | Deposit date: | 2012-11-19 | Release date: | 2013-04-03 | Method: | X-RAY DIFFRACTION (1.6 Å) | Cite: | Structural and functional analysis of the CspB protease required for Clostridium spore germination. Plos Pathog., 9, 2013
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3PA8
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![BU of 3pa8 by Molmil](/molmil-images/mine/3pa8) | |
5Z1W
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6MW4
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![BU of 6mw4 by Molmil](/molmil-images/mine/6mw4) | |
6PSL
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![BU of 6psl by Molmil](/molmil-images/mine/6psl) | Structure of a N-Me-D-Gln4,D-aza-Thr8,Arg10-teixobactin analogue | Descriptor: | CHLORIDE ION, teixobactin analogue | Authors: | Nowick, J.S, Yang, H, Pishenko, A, Li, X. | Deposit date: | 2019-07-12 | Release date: | 2019-11-27 | Last modified: | 2023-11-15 | Method: | X-RAY DIFFRACTION (2.1 Å) | Cite: | Design, Synthesis, and Study of Lactam and Ring-Expanded Analogues of Teixobactin. J.Org.Chem., 85, 2020
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6DBD
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![BU of 6dbd by Molmil](/molmil-images/mine/6dbd) | Crystal Structure of VHH R326 | Descriptor: | ACETATE ION, SODIUM ION, nanobody VHH R326 | Authors: | Brooks, C.L, Toride King, M, Huh, I. | Deposit date: | 2018-05-03 | Release date: | 2018-07-18 | Last modified: | 2023-10-04 | Method: | X-RAY DIFFRACTION (1.755 Å) | Cite: | Structural basis of VHH-mediated neutralization of the food-borne pathogenListeria monocytogenes. J. Biol. Chem., 293, 2018
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6DBA
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![BU of 6dba by Molmil](/molmil-images/mine/6dba) | Crystal Structure of VHH R303 | Descriptor: | nanobody VHH R303 | Authors: | Brooks, C.L, Toride King, M, Huh, I. | Deposit date: | 2018-05-02 | Release date: | 2018-07-18 | Last modified: | 2023-10-04 | Method: | X-RAY DIFFRACTION (1.3 Å) | Cite: | Structural basis of VHH-mediated neutralization of the food-borne pathogenListeria monocytogenes. J. Biol. Chem., 293, 2018
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6DBE
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![BU of 6dbe by Molmil](/molmil-images/mine/6dbe) | Crystal Structure of VHH R330 | Descriptor: | 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, nanobody VHH R303 | Authors: | Brooks, C.L, Toride King, M, Huh, I. | Deposit date: | 2018-05-03 | Release date: | 2018-07-18 | Last modified: | 2023-10-04 | Method: | X-RAY DIFFRACTION (1.65 Å) | Cite: | Structural basis of VHH-mediated neutralization of the food-borne pathogenListeria monocytogenes. J. Biol. Chem., 293, 2018
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6DBF
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6DBG
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![BU of 6dbg by Molmil](/molmil-images/mine/6dbg) | |