3PA8
Structure of the C. difficile TcdB cysteine protease domain in complex with a peptide inhibitor
Summary for 3PA8
Entry DOI | 10.2210/pdb3pa8/pdb |
Related PRD ID | PRD_000971 |
Descriptor | Toxin B, N-acetylglycyl-N-[(3S)-1-hydroxy-5-methyl-2-oxohexan-3-yl]-L-serinamide, CALCIUM ION, ... (6 entities in total) |
Functional Keywords | clan cd cysteine protease, protease, toxin, toxin-peptide inhibitor complex, toxin/peptide inhibitor |
Biological source | Clostridium difficile |
Total number of polymer chains | 2 |
Total formula weight | 59877.68 |
Authors | Lupardus, P.J.,Garcia, K.C. (deposition date: 2010-10-18, release date: 2010-12-15, Last modification date: 2023-09-06) |
Primary citation | Puri, A.W.,Lupardus, P.J.,Deu, E.,Albrow, V.E.,Garcia, K.C.,Bogyo, M.,Shen, A. Rational design of inhibitors and activity-based probes targeting Clostridium difficile virulence factor TcdB. Chem.Biol., 17:1201-1211, 2010 Cited by PubMed: 21095570DOI: 10.1016/j.chembiol.2010.09.011 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2 Å) |
Structure validation
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