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5CFS

Crystal Structure of ANT(2")-Ia in complex with AMPCPP and tobramycin

Summary for 5CFS
Entry DOI10.2210/pdb5cfs/pdb
Related4XJE 5CFT 5CFU
DescriptorAAD(2''),Gentamicin 2''-nucleotidyltransferase,Gentamicin resistance protein, MANGANESE (II) ION, TOBRAMYCIN, ... (7 entities in total)
Functional Keywordsantibiotic resistance, nucleotidyltransferase, ampcpp, tobramycin, rossmann fold, transferase-antibiotic complex, transferase/antibiotic
Biological sourcePseudomonas aeruginosa
Total number of polymer chains1
Total formula weight22449.59
Authors
Rodionov, D.,Bassenden, A.V.,Berghuis, A.M. (deposition date: 2015-07-08, release date: 2016-03-16, Last modification date: 2023-09-27)
Primary citationBassenden, A.V.,Rodionov, D.,Shi, K.,Berghuis, A.M.
Structural Analysis of the Tobramycin and Gentamicin Clinical Resistome Reveals Limitations for Next-generation Aminoglycoside Design.
Acs Chem.Biol., 11:1339-1346, 2016
Cited by
PubMed: 26900880
DOI: 10.1021/acschembio.5b01070
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.7 Å)
Structure validation

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