1P8J
CRYSTAL STRUCTURE OF THE PROPROTEIN CONVERTASE FURIN
Summary for 1P8J
Entry DOI | 10.2210/pdb1p8j/pdb |
Related PRD ID | PRD_000278 |
Descriptor | Furin precursor, DECANOYL-ARG-VAL-LYS-ARG-CHLOROMETHYLKETONE INHIBITOR, beta-D-galactopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-[beta-D-galactopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)]alpha-D-mannopyranose-(1-3)-[2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-6)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[beta-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ... (8 entities in total) |
Functional Keywords | prohormone convertase, spc1, pace, p-domain, chloromethylketone, hydrolase-hydrolase inhibitor complex, hydrolase/hydrolase inhibitor |
Biological source | Mus musculus (house mouse) More |
Total number of polymer chains | 16 |
Total formula weight | 426622.72 |
Authors | Henrich, S.,Cameron, A.,Bourenkov, G.P.,Kiefersauer, R.,Huber, R.,Lindberg, I.,Bode, W.,Than, M.E. (deposition date: 2003-05-07, release date: 2003-07-08, Last modification date: 2020-07-29) |
Primary citation | Henrich, S.,Cameron, A.,Bourenkov, G.P.,Kiefersauer, R.,Huber, R.,Lindberg, I.,Bode, W.,Than, M.E. The Crystal Structure of the Proprotein Processing Proteinase Furin Explains its Stringent Specificity Nat.Struct.Biol., 10:520-526, 2003 Cited by PubMed: 12794637DOI: 10.1038/nsb941 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.6 Å) |
Structure validation
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