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9XBU

Crystal structure of human SIRT5 in XR-0931

This is a non-PDB format compatible entry.
Summary for 9XBU
Entry DOI10.2210/pdb9xbu/pdb
DescriptorNAD-dependent protein deacylase sirtuin-5, mitochondrial, ZINC ION, 3-[[(~{Z})-~{N}'-cyano-~{N}-[3-[[2-(6-ethoxypyridin-3-yl)-5-[[4-(trifluoromethyloxy)phenyl]methylcarbamoyl]pyrimidin-4-yl]amino]propyl]carbamimidoyl]amino]propanoic acid, ... (4 entities in total)
Functional Keywordssirt5, hydrolase, hydrolase inhibitor
Biological sourceHomo sapiens (human)
Total number of polymer chains2
Total formula weight59954.78
Authors
Xiong, R. (deposition date: 2025-10-24, release date: 2026-10-28)
Primary citationXiong, R.,yang, L.L.
Crystal structure of human SIRT5 in XR-0931
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.242 Å)
Structure validation

262513

PDB entries from 2026-11-04

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