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9QOB

CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 IN COMPLEX with compound 4

This is a non-PDB format compatible entry.
Summary for 9QOB
Entry DOI10.2210/pdb9qob/pdb
DescriptorBromodomain-containing protein 4, 1,2-ETHANEDIOL, (5-phenyl-[1,3]thiazolo[2,3-c][1,2,4]triazol-3-yl)methanol, ... (4 entities in total)
Functional Keywordsbromodomain-containing protein 4 isoform long, brd4, bromodomain-containing protein 4, cap, hunk1, mcap, mitotic chromosome associated protein, cell cycle
Biological sourceHomo sapiens (human)
Total number of polymer chains1
Total formula weight15367.71
Authors
Primary citationKrojer, T.,Martinez-Cartro, M.,Picaud, S.,Filippakopoulos, P.,Arrowsmith, C.H.,Edwards, A.M.,Bountra, C.,Barril, X.,von Delft, F.
CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 IN COMPLEX with compound 2
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.37 Å)
Structure validation

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