9OU2
K-Ras Wild Type 1-169 Bound to BI-2865 at 100 K
Summary for 9OU2
| Entry DOI | 10.2210/pdb9ou2/pdb |
| Descriptor | GTPase KRas, MAGNESIUM ION, (4S)-2-azanyl-4-methyl-4-[3-[4-[(1S)-1-[(2S)-1-methylpyrrolidin-1-ium-2-yl]ethoxy]pyrimidin-2-yl]-1,2,4-oxadiazol-5-yl]-6,7-dihydro-5H-1-benzothiophene-3-carbonitrile, ... (5 entities in total) |
| Functional Keywords | gtpase, hydrolase |
| Biological source | Homo sapiens (human) |
| Total number of polymer chains | 1 |
| Total formula weight | 20205.85 |
| Authors | Xu, M.,Deck, S.L.,Milano, S.K.,Cerione, R.A. (deposition date: 2025-05-28, release date: 2026-06-17) |
| Primary citation | Xu, M.,Deck, S.L.,Milano, S.K.,Cerione, R.A. Oncogenic K-Ras Mutants Bound to Inhibitors To Be Published, |
| Experimental method | X-RAY DIFFRACTION (1.55 Å) |
Structure validation
Download full validation report






