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9OU2

K-Ras Wild Type 1-169 Bound to BI-2865 at 100 K

Summary for 9OU2
Entry DOI10.2210/pdb9ou2/pdb
DescriptorGTPase KRas, MAGNESIUM ION, (4S)-2-azanyl-4-methyl-4-[3-[4-[(1S)-1-[(2S)-1-methylpyrrolidin-1-ium-2-yl]ethoxy]pyrimidin-2-yl]-1,2,4-oxadiazol-5-yl]-6,7-dihydro-5H-1-benzothiophene-3-carbonitrile, ... (5 entities in total)
Functional Keywordsgtpase, hydrolase
Biological sourceHomo sapiens (human)
Total number of polymer chains1
Total formula weight20205.85
Authors
Xu, M.,Deck, S.L.,Milano, S.K.,Cerione, R.A. (deposition date: 2025-05-28, release date: 2026-06-17)
Primary citationXu, M.,Deck, S.L.,Milano, S.K.,Cerione, R.A.
Oncogenic K-Ras Mutants Bound to Inhibitors
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.55 Å)
Structure validation

255239

PDB entries from 2026-06-17

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