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9I0A

CARM1 in complex with arg-aDMA analog

This is a non-PDB format compatible entry.
Summary for 9I0A
Entry DOI10.2210/pdb9i0a/pdb
DescriptorHistone-arginine methyltransferase CARM1, (phenylmethyl) (2S)-5-[[N-[3-[(2R,3S,4R,5R)-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]propyl]-N-methyl-carbamimidoyl]amino]-2-(phenylmethoxycarbonylamino)pentanoate (3 entities in total)
Functional Keywordsprotein arginine n-methyltransferase, prmt, carm1, transition state mimics, transcription, transferase
Biological sourceMus musculus (house mouse)
Total number of polymer chains4
Total formula weight166160.87
Authors
Cura, V.,Dursun, E.,Troffer, N.,Cavarelli, J. (deposition date: 2025-01-14, release date: 2026-01-28)
Primary citationCura, V.,Dursun, E.,Troffer, N.,Cavarelli, J.
CARM1 in complex with arg-aDMA analog
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.22 Å)
Structure validation

251422

PDB entries from 2026-04-01

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