9BFM
Cryo-EM co-structure of AcrB with the EPM35 efflux pump inhibitor
This is a non-PDB format compatible entry.
Summary for 9BFM
Entry DOI | 10.2210/pdb9bfm/pdb |
EMDB information | 44500 |
Descriptor | Multidrug efflux pump subunit AcrB, (2S)-1-(3,4-dichlorophenoxy)-3-(4-{[4-(trifluoromethyl)pyrimidin-2-yl]amino}piperidin-1-yl)propan-2-ol (3 entities in total) |
Functional Keywords | acrb multidrug efflux pump, translocase |
Biological source | Escherichia coli K-12 |
Total number of polymer chains | 3 |
Total formula weight | 341460.84 |
Authors | |
Primary citation | Allgood, S.C.,Su, C.C.,Crooks, A.L.,Meyer, C.T.,Zhou, B.,Betterton, M.D.,Barbachyn, M.R.,Yu, E.W.,Detweiler, C.S. Bacterial efflux pump modulators prevent bacterial growth in macrophages and under broth conditions that mimic the host environment. mBio, 14:e0249223-, 2023 Cited by PubMed: 37921493DOI: 10.1073/pnas.1901346116 PDB entries with the same primary citation |
Experimental method | ELECTRON MICROSCOPY (2.71 Å) |
Structure validation
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