9LUS

Structure of human G9a SET-domain in complex with FLAV27 inhibitor

This is a non-PDB format compatible entry.

Summary for 9LUS

• Entry DOI: 10.2210/pdb9lus/pdb
• Related: 7t7l
• Descriptor: Histone-lysine N-methyltransferase EHMT2, ZINC ION, 3-[1-[[(2~{S})-4-(phenylmethyl)-1,4-oxazepan-2-yl]methyl]piperidin-4-yl]phenol, ... (4 entities in total)
• Functional Keywords: histone, complex, set domain, transferase, transferase-inhibitor complex, transferase/inhibitor
• Biological source: Homo sapiens (human)
• Total number of polymer chains: 2
• Total formula weight: 69879.88

Authors

Singh, R.K.,Dai, S. (deposition date: 2025-02-10, release date: 2026-02-18)

• Primary citation: Singh, R.K.,Dai, S.; Structure of human G9a SET-domain in complex with FLAV27 inhibitor; To Be Published,

Experimental method

X-RAY DIFFRACTION (2.7 Å)