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8WJY

PKMYT1_Cocrystal_Cpd 4

Summary for 8WJY
Entry DOI10.2210/pdb8wjy/pdb
DescriptorMembrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase, [6-azanyl-5-(2,6-dimethyl-3-oxidanyl-phenyl)-2,3-dimethyl-pyrrolo[2,3-b]pyrazin-7-yl]-(6,7-dihydro-4~{H}-pyrazolo[1,5-a]pyrazin-5-yl)methanone, DIMETHYL SULFOXIDE, ... (5 entities in total)
Functional Keywordsinhibitor, co-crystal, antitumor protein
Biological sourceHomo sapiens (human)
Total number of polymer chains1
Total formula weight35099.85
Authors
Wang, Y.,Wang, C.,Liu, T.,Qi, H.,Chen, S.,Cai, X.,Zhang, M.,Aliper, A.,Ren, F.,Ding, X.,Zhavoronkov, A. (deposition date: 2023-09-26, release date: 2023-11-22)
Primary citationWang, Y.,Wang, C.,Liu, T.,Qi, H.,Chen, S.,Cai, X.,Zhang, M.,Aliper, A.,Ren, F.,Ding, X.,Zhavoronkov, A.
PKMYT1_Cocrystal_Cpd 4
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.88 Å)
Structure validation

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