8SIF
Crystal structure of Escherichia coli HPPK in complex with bisubstrate inhibitor HP-101
Summary for 8SIF
Entry DOI | 10.2210/pdb8sif/pdb |
Descriptor | 2-amino-4-hydroxy-6-hydroxymethyldihydropteridine pyrophosphokinase, 5'-S-{(2R,4R)-1-[3-(2-amino-4-oxo-4,7-dihydro-3H-pyrrolo[2,3-d]pyrimidin-5-yl)propyl]-2-carboxypiperidin-4-yl}-5'-thioadenosine (3 entities in total) |
Functional Keywords | hppk, bisubstrate inhibitor, hp-101, transferase, transferase-inhibitor complex, transferase/inhibitor |
Biological source | Escherichia coli |
Total number of polymer chains | 1 |
Total formula weight | 18698.38 |
Authors | |
Primary citation | Shi, G.,Shaw, G.X.,Ji, X. The first bisubstrate inhibitor of HPPK exhibiting cell permeability To be published, |
Experimental method | X-RAY DIFFRACTION (1.7 Å) |
Structure validation
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