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8R18

Pim1 in complex with (E)-4-(4-hydroxystyryl)benzoic acid and Pimtide

Summary for 8R18
Entry DOI10.2210/pdb8r18/pdb
Related7QB2 7QFM 7Z6U 8AFR 8R0H 8R0Q 8R0W 8R0Y 8R10
DescriptorSerine/threonine-protein kinase pim-1, Pimtide, GLYCEROL, ... (6 entities in total)
Functional Keywordsserine kinase, kinase, complex, pim1, pim, pim-1, inhibitor, tumorigenisis, cancer, pimtide, proto oncogen, atp, phosphorylation, apoptosis, cell cycle, transferase
Biological sourceHomo sapiens (human)
More
Total number of polymer chains2
Total formula weight37657.74
Authors
Hochban, P.M.M.,Heine, A.,Diederich, W.E. (deposition date: 2023-11-01, release date: 2024-03-20)
Primary citationHochban, P.M.M.,Heyder, L.,Heine, A.,Diederich, W.E.
Pim1 in complex with (E)-4-(4-hydroxystyryl)benzoic acid and Pimtide
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.89 Å)
Structure validation

218853

PDB entries from 2024-04-24

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