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8R10

Pim1 in complex with 4-(4-hydroxystyryl)benzoic acid and Pimtide

Summary for 8R10
Entry DOI10.2210/pdb8r10/pdb
Related7QB2 7QFM 7Z6U 8AFR 8R0H 8R0Q 8R0W 8R0Y
DescriptorSerine/threonine-protein kinase pim-1, Pimtide, (Z)-4-(4-hydroxystyryl)benzoic acid, ... (4 entities in total)
Functional Keywordsserine kinase, kinase, complex, pim1, pim, pim-1, inhibitor, tumorigenisis, cancer, pimtide, proto oncogen, atp, phosphorylation, apoptosis, cell cycle, transferase
Biological sourceHomo sapiens (human)
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Total number of polymer chains2
Total formula weight37503.58
Authors
Hochban, P.M.M.,Heine, A.,Diederich, W.E. (deposition date: 2023-11-01, release date: 2024-03-20)
Primary citationHochban, P.M.M.,Heyder, L.,Heine, A.,Diederich, W.E.
Pim1 in complex with 4-(4-hydroxystyryl)benzoic acid and Pimtide
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.2 Å)
Structure validation

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PDB entries from 2024-04-24

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