8R0Y
Pim1 in complex with 3-((3-hydroxyphenyl)amino)quinoxaline-2-carboxylic acid and Pimtide
Summary for 8R0Y
| Entry DOI | 10.2210/pdb8r0y/pdb |
| Related | 7QB2 7QFM 7Z6U 8AFR 8R0H 8R0Q 8R0W |
| Descriptor | Serine/threonine-protein kinase pim-1, Pimtide, GLYCEROL, ... (5 entities in total) |
| Functional Keywords | serine kinase, kinase, complex, pim1, pim, pim-1, inhibitor, tumorigenisis, cancer, pimtide, proto oncogen, atp, phosphorylation, apoptosis, cell cycle, transferase |
| Biological source | Homo sapiens (human) More |
| Total number of polymer chains | 2 |
| Total formula weight | 37636.69 |
| Authors | |
| Primary citation | Hochban, P.M.M.,Daude, M.,Heine, A.,Diederich, W.E. Pim1 in complex with 3-((3-hydroxyphenyl)amino)quinoxaline-2-carboxylic acid and Pimtide To Be Published, |
| Experimental method | X-RAY DIFFRACTION (2.05 Å) |
Structure validation
Download full validation report






