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8R0W

Pim1 in complex with 5-bromobenzo[d]oxazol-2-amine and Pimtide

Summary for 8R0W
Entry DOI10.2210/pdb8r0w/pdb
Related7QB2 7QFM 7Z6U 8AFR 8R0H 8R0Q
DescriptorSerine/threonine-protein kinase pim-1, Pimtide, 1,2-ETHANEDIOL, ... (6 entities in total)
Functional Keywordsserine kinase, kinase, complex, pim1, pim, pim-1, inhibitor, tumorigenisis, cancer, pimtide, proto oncogen, atp, phosphorylation, apoptosis, cell cycle, transferase
Biological sourceHomo sapiens (human)
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Total number of polymer chains2
Total formula weight37814.71
Authors
Hochban, P.M.M.,Heine, A.,Diederich, W.E. (deposition date: 2023-11-01, release date: 2024-11-13)
Primary citationHochban, P.M.M.,Daude, M.,Heine, A.,Diederich, W.E.
Pim1 in complex with 5-bromobenzo[d]oxazol-2-amine and Pimtide
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.95 Å)
Structure validation

248942

PDB entries from 2026-02-11

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