8R0W
Pim1 in complex with 5-bromobenzo[d]oxazol-2-amine and Pimtide
Summary for 8R0W
| Entry DOI | 10.2210/pdb8r0w/pdb |
| Related | 7QB2 7QFM 7Z6U 8AFR 8R0H 8R0Q |
| Descriptor | Serine/threonine-protein kinase pim-1, Pimtide, 1,2-ETHANEDIOL, ... (6 entities in total) |
| Functional Keywords | serine kinase, kinase, complex, pim1, pim, pim-1, inhibitor, tumorigenisis, cancer, pimtide, proto oncogen, atp, phosphorylation, apoptosis, cell cycle, transferase |
| Biological source | Homo sapiens (human) More |
| Total number of polymer chains | 2 |
| Total formula weight | 37814.71 |
| Authors | |
| Primary citation | Hochban, P.M.M.,Daude, M.,Heine, A.,Diederich, W.E. Pim1 in complex with 5-bromobenzo[d]oxazol-2-amine and Pimtide To Be Published, |
| Experimental method | X-RAY DIFFRACTION (1.95 Å) |
Structure validation
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