8JVJ
Structure of human TRPV4 with antagonist A2 and RhoA
Summary for 8JVJ
Entry DOI | 10.2210/pdb8jvj/pdb |
EMDB information | 36676 |
Descriptor | Transient receptor potential cation channel subfamily V member 4,3C-GFP, Transforming protein RhoA, [6-[[4-(2,4-dimethyl-1,3-thiazol-5-yl)-1,3-thiazol-2-yl]amino]pyridin-3-yl]-[(1~{S},5~{R})-3-[5-(trifluoromethyl)pyrimidin-2-yl]-3,8-diazabicyclo[3.2.1]octan-8-yl]methanone (3 entities in total) |
Functional Keywords | channel, membrane protein |
Biological source | Homo sapiens (human) More |
Total number of polymer chains | 8 |
Total formula weight | 604001.33 |
Authors | |
Primary citation | Fan, J.,Guo, C.,Liao, D.,Ke, H.,Lei, J.,Xie, W.,Tang, Y.,Tominaga, M.,Huang, Z.,Lei, X. Structural Pharmacology of TRPV4 Antagonists. Adv Sci, 11:e2401583-e2401583, 2024 Cited by PubMed: 38659239DOI: 10.1002/advs.202401583 PDB entries with the same primary citation |
Experimental method | ELECTRON MICROSCOPY (3.44 Å) |
Structure validation
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