8JU5
Structure of human TRPV4 with antagonist A1
Summary for 8JU5
Entry DOI | 10.2210/pdb8ju5/pdb |
EMDB information | 36659 |
Descriptor | Transient receptor potential cation channel subfamily V member 4,3C-GFP, 4-[(3~{S},4~{S})-4-(aminomethyl)-1-(5-chloranylpyridin-2-yl)sulfonyl-4-oxidanyl-pyrrolidin-3-yl]oxy-2-fluoranyl-benzenecarbonitrile (2 entities in total) |
Functional Keywords | channel, membrane protein |
Biological source | Homo sapiens (human) More |
Total number of polymer chains | 4 |
Total formula weight | 515367.89 |
Authors | |
Primary citation | Fan, J.,Guo, C.,Liao, D.,Ke, H.,Lei, J.,Xie, W.,Tang, Y.,Tominaga, M.,Huang, Z.,Lei, X. Structural Pharmacology of TRPV4 Antagonists. Adv Sci, 11:e2401583-e2401583, 2024 Cited by PubMed: 38659239DOI: 10.1002/advs.202401583 PDB entries with the same primary citation |
Experimental method | ELECTRON MICROSCOPY (3.74 Å) |
Structure validation
Download full validation report