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8HLR

Human ADP-ribosyltransferase 1 (PARP1) catalytic domain bound to Fluzoparib (SHR3162)

Summary for 8HLR
Entry DOI10.2210/pdb8hlr/pdb
DescriptorPoly [ADP-ribose] polymerase 1, processed C-terminus, Fluzoparib, SULFATE ION, ... (4 entities in total)
Functional Keywordsdna adp-ribosyltransferase 1, parp1, fluzoparib, shr3162, transferase
Biological sourceHomo sapiens (Human)
Total number of polymer chains2
Total formula weight81208.09
Authors
Wang, X.Y.,Zhou, J.,Xu, B.L. (deposition date: 2022-11-30, release date: 2024-05-01)
Primary citationWang, X.Y.,Zhou, J.,Xu, B.L.
Human ADP-ribosyltransferase 1 (PARP1) catalytic domain bound to Fluzoparib (SHR3162)
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.85 Å)
Structure validation

220113

PDB entries from 2024-05-22

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