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8BZS

The crystal structure of glycogen phosphorylase in complex with baicalein

Summary for 8BZS
Entry DOI10.2210/pdb8bzs/pdb
DescriptorGlycogen phosphorylase, muscle form, PYRIDOXAL-5'-PHOSPHATE, 5,6,7-trihydroxy-2-phenyl-4H-chromen-4-one, ... (4 entities in total)
Functional Keywordstransferase
Biological sourceOryctolagus cuniculus (rabbit)
Total number of polymer chains1
Total formula weight97939.78
Authors
Koulas, S.M.,Mathomes, R.,Hayes, J.M.,Leonidas, D.D. (deposition date: 2022-12-15, release date: 2023-09-13)
Primary citationMathomes, R.T.,Koulas, S.M.,Tsialtas, I.,Stravodimos, G.,Welsby, P.J.,Psarra, A.G.,Stasik, I.,Leonidas, D.D.,Hayes, J.M.
Multidisciplinary docking, kinetics and X-ray crystallography studies of baicalein acting as a glycogen phosphorylase inhibitor and determination of its' potential against glioblastoma in cellular models.
Chem.Biol.Interact., 382:110568-110568, 2023
Cited by
PubMed: 37277066
DOI: 10.1016/j.cbi.2023.110568
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.25 Å)
Structure validation

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