Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

8B6M

Tankyrase 2 in complex with an inhibitor

Summary for 8B6M
Entry DOI10.2210/pdb8b6m/pdb
DescriptorPoly [ADP-ribose] polymerase tankyrase-2, ~{N}-(2-methoxyphenyl)-4-[[2-(4-oxidanylidene-3~{H}-quinazolin-2-yl)ethyl-(thiophen-2-ylmethyl)carbamoyl]amino]benzamide, SULFATE ION, ... (7 entities in total)
Functional Keywordsinhibitor, transferase
Biological sourceHomo sapiens (human)
More
Total number of polymer chains4
Total formula weight51406.61
Authors
Bosetti, C.,Sowa, S.T.,Lehtio, L. (deposition date: 2022-09-27, release date: 2023-10-11)
Primary citationBosetti, C.,Sowa, S.T.,Lehtio, L.
Tankyrase 2 in complex with an inhibitor
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.6 Å)
Structure validation

218853

PDB entries from 2024-04-24

PDB statisticsPDBj update infoContact PDBjnumon