8B6M

Tankyrase 2 in complex with an inhibitor

Summary for 8B6M

• Entry DOI: 10.2210/pdb8b6m/pdb
• Descriptor: Poly [ADP-ribose] polymerase tankyrase-2, ~{N}-(2-methoxyphenyl)-4-[[2-(4-oxidanylidene-3~{H}-quinazolin-2-yl)ethyl-(thiophen-2-ylmethyl)carbamoyl]amino]benzamide, SULFATE ION, ... (7 entities in total)
• Functional Keywords: inhibitor, transferase
• Biological source: Homo sapiens (human); More
• Total number of polymer chains: 4
• Total formula weight: 51406.61

Authors

Bosetti, C.,Sowa, S.T.,Lehtio, L. (deposition date: 2022-09-27, release date: 2023-10-11)

• Primary citation: Bosetti, C.,Sowa, S.T.,Lehtio, L.; Tankyrase 2 in complex with an inhibitor; To Be Published,

Experimental method

X-RAY DIFFRACTION (1.6 Å)