Summary for 8YKI
Entry DOI | 10.2210/pdb8yki/pdb |
Descriptor | Fibroblast growth factor receptor 1, Tasurgratinib, CHLORIDE ION, ... (4 entities in total) |
Functional Keywords | fgf receptor kinase, proteros biostructures gmbh, transferase |
Biological source | Homo sapiens (human) |
Total number of polymer chains | 2 |
Total formula weight | 73479.18 |
Authors | |
Primary citation | Kawano, S.,Kawada, M.I.,Fukushima, S.,Arai, Y.,Shibata, T.,Miyano, S.W. Antitumor Activity of Tasurgratinib as an Orally Available FGFR1-3 Inhibitor in Cholangiocarcinoma Models With FGFR2-fusion. Anticancer Res., 44:2393-2406, 2024 Cited by PubMed: 38821585DOI: 10.21873/anticanres.17046 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.79 Å) |
Structure validation
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