8WSM
NLRP3 NACHT domain in complex with compound 32
Summary for 8WSM
Entry DOI | 10.2210/pdb8wsm/pdb |
Descriptor | NACHT, LRR and PYD domains-containing protein 3, MAGNESIUM ION, ADENOSINE-5'-DIPHOSPHATE, ... (5 entities in total) |
Functional Keywords | inflammasome, immune system |
Biological source | Homo sapiens (human) |
Total number of polymer chains | 1 |
Total formula weight | 65056.23 |
Authors | Akai, S.,Orita, T.,Adachi, T. (deposition date: 2023-10-17, release date: 2023-11-22, Last modification date: 2024-01-03) |
Primary citation | Ohba, Y.,Adachi, K.,Furukawa, T.,Nishimaru, T.,Sakurai, K.,Masuo, R.,Inami, T.,Orita, T.,Akai, S.,Adachi, T.,Usui, K.,Hamada, Y.,Mori, M.,Kurimoto, T.,Wakashima, T.,Akiyama, Y.,Miyazaki, S.,Noji, S. Discovery of Novel NLRP3 Inflammasome Inhibitors Composed of an Oxazole Scaffold Bearing an Acylsulfamide. Acs Med.Chem.Lett., 14:1833-1838, 2023 Cited by PubMed: 38116417DOI: 10.1021/acsmedchemlett.3c00433 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.7 Å) |
Structure validation
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