8WPG
Human calcium-sensing receptor bound with cinacalcet in detergent
Summary for 8WPG
Entry DOI | 10.2210/pdb8wpg/pdb |
EMDB information | 37716 |
Descriptor | Extracellular calcium-sensing receptor, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose, ... (7 entities in total) |
Functional Keywords | gpcr, allosteric modulator, activation, dimeric, membrane protein |
Biological source | Homo sapiens (human) |
Total number of polymer chains | 2 |
Total formula weight | 208360.58 |
Authors | Ling, S.L.,Meng, X.Y.,Tian, C.L. (deposition date: 2023-10-10, release date: 2023-11-22, Last modification date: 2024-02-21) |
Primary citation | Ling, S.,Meng, X.,Zhang, Y.,Xia, Z.,Zhou, Y.,Yang, F.,Shi, P.,Shi, C.,Tian, C. Structural insights into asymmetric activation of the calcium-sensing receptor-G q complex. Cell Res., 34:169-172, 2024 Cited by PubMed: 37919470DOI: 10.1038/s41422-023-00892-2 PDB entries with the same primary citation |
Experimental method | ELECTRON MICROSCOPY (2.7 Å) |
Structure validation
Download full validation report