7ZM2
Crystal structure of HsaD from Mycobacterium tuberculosis in complex with Cyclophostin-like inhibitor CyC8b
Summary for 7ZM2
Entry DOI | 10.2210/pdb7zm2/pdb |
Related | 7ZJT 7ZM1 |
Descriptor | 4,5:9,10-diseco-3-hydroxy-5,9,17-trioxoandrosta-1(10),2-diene-4-oate hydrolase, methoxy-[(3~{R})-3-[(2~{R})-1-methoxy-1,3-bis(oxidanylidene)butan-2-yl]pentadecyl]phosphinic acid, SULFATE ION, ... (4 entities in total) |
Functional Keywords | hsad, m. tuberculosis, cholesterol, inhibitor, hydrolase |
Biological source | Mycobacterium tuberculosis H37Rv |
Total number of polymer chains | 2 |
Total formula weight | 67294.54 |
Authors | Barelier, S.,Roig-Zamboni, V.,Cavalier, J.F.,Sulzenbacher, G. (deposition date: 2022-04-19, release date: 2022-09-28, Last modification date: 2024-02-07) |
Primary citation | Barelier, S.,Avellan, R.,Gnawali, G.R.,Fourquet, P.,Roig-Zamboni, V.,Poncin, I.,Point, V.,Bourne, Y.,Audebert, S.,Camoin, L.,Spilling, C.D.,Canaan, S.,Cavalier, J.F.,Sulzenbacher, G. Direct capture, inhibition and crystal structure of HsaD (Rv3569c) from M. tuberculosis. Febs J., 290:1563-1582, 2023 Cited by PubMed: 36197115DOI: 10.1111/febs.16645 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.2 Å) |
Structure validation
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