7Z2P
Tubulin-nocodazole complex
Summary for 7Z2P
Entry DOI | 10.2210/pdb7z2p/pdb |
Descriptor | Tubulin alpha-1B chain, PHOSPHOMETHYLPHOSPHONIC ACID ADENYLATE ESTER, Tubulin beta-2B chain, ... (11 entities in total) |
Functional Keywords | tubulin fold, cytoskeleton, microtubule, cell cycle |
Biological source | Rattus norvegicus (Norway rat) More |
Total number of polymer chains | 6 |
Total formula weight | 265183.93 |
Authors | Prota, A.E.,Muehlethaler, T.,Cavalli, A.,Steinmetz, M.O. (deposition date: 2022-02-28, release date: 2022-08-31, Last modification date: 2024-01-31) |
Primary citation | de la Roche, N.M.,Muhlethaler, T.,Di Martino, R.M.C.,Ortega, J.A.,Gioia, D.,Roy, B.,Prota, A.E.,Steinmetz, M.O.,Cavalli, A. Novel fragment-derived colchicine-site binders as microtubule-destabilizing agents. Eur.J.Med.Chem., 241:114614-114614, 2022 Cited by PubMed: 35939994DOI: 10.1016/j.ejmech.2022.114614 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2 Å) |
Structure validation
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