7X3P
Crystal structure of human SIRT5 in complex with diazirine inhibitor 9
7X3P の概要
エントリーDOI | 10.2210/pdb7x3p/pdb |
分子名称 | NAD-dependent protein deacylase sirtuin-5, mitochondrial, 5-[[(5~{S})-6-[[(1~{S})-1-(4-hydroxyphenyl)-2-oxidanylidene-2-(prop-2-ynylamino)ethyl]amino]-6-oxidanylidene-5-[[4-[3-(trifluoromethyl)-1,2-diazirin-3-yl]phenyl]carbonylamino]hexyl]amino]-5-sulfanylidene-pentanoic acid, DI(HYDROXYETHYL)ETHER, ... (5 entities in total) |
機能のキーワード | inhibitor, complex, hydrolase, hydrolase-hydrolase inhibitor complex, hydrolase/hydrolase inhibitor |
由来する生物種 | Homo sapiens (human) |
タンパク質・核酸の鎖数 | 1 |
化学式量合計 | 31029.54 |
構造登録者 | |
主引用文献 | Li, G.-B.,Deng, J. Crystal structure of human SIRT5 in complex with diazirine inhibitor 9 To Be Published, |
実験手法 | X-RAY DIFFRACTION (1.56 Å) |
構造検証レポート
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