7TV9
HUMAN COMPLEMENT COMPONENT C3B IN COMPLEX WITH APL-1030
Summary for 7TV9
Entry DOI | 10.2210/pdb7tv9/pdb |
Descriptor | Complement C3 beta chain, Complement C3b alpha' chain, APL-1030 Nanofitin, ... (5 entities in total) |
Functional Keywords | immune system, complement protein complex |
Biological source | synthetic construct More |
Total number of polymer chains | 3 |
Total formula weight | 183655.56 |
Authors | Fontano, E.,Nadupalli, A.,Lakshminarasimhan, D.,White, A.,Garlish, J.,Cinier, M.,Chevrel, A.,Perrocheau, A.,Eyerman, D.,Orme, M.,Kitten, O.,Scheibler, L. (deposition date: 2022-02-04, release date: 2022-03-30, Last modification date: 2023-10-18) |
Primary citation | Garlich, J.,Cinier, M.,Chevrel, A.,Perrocheau, A.,Eyerman, D.J.,Orme, M.,Kitten, O.,Scheibler, L. Discovery of APL-1030, a Novel, High-Affinity Nanofitin Inhibitor of C3-Mediated Complement Activation. Biomolecules, 12:-, 2022 Cited by PubMed: 35327625DOI: 10.3390/biom12030432 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (3.4 Å) |
Structure validation
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