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7S6U

Leishmania infantum Glycogen Synthase Kinase 3 beta bound to AZD5438

Summary for 7S6U
Entry DOI10.2210/pdb7s6u/pdb
DescriptorGlycogen synthase kinase 3, 4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{N}-(4-methylsulfonylphenyl)pyrimidin-2-amine, 1,2-ETHANEDIOL, ... (5 entities in total)
Functional Keywordsprotein kinase, inhibitor, transferase, gsk3s, gsk3beta, leishmania infantum, transferase-inhibitor complex, transferase/inhibitor
Biological sourceLeishmania infantum
Total number of polymer chains1
Total formula weight41628.51
Authors
dos Reis, C.V.,Ramos, P.Z.,Counago, R.M. (deposition date: 2021-09-15, release date: 2022-11-09, Last modification date: 2023-11-15)
Primary citationRamos, P.Z.,dos Reis, C.V.,Counago, R.M.
Leishmania infantum Glycogen Synthase Kinase 3 beta bound to AZD5438
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.74 Å)
Structure validation

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