7NGW
Mycobacterium tuberculosis transcriptional regulator EthR with bound inhibitory compound
Summary for 7NGW
Entry DOI | 10.2210/pdb7ngw/pdb |
Related | 5NGD 5NGG 5NGI 5NGJ 5NGK 5NGM 5NGN 5NGO 5NGR 5NGS 5NGT 5NGU |
Descriptor | HTH-type transcriptional regulator EthR, ~{N}-(4-hydroxyphenyl)-4-methyl-piperidine-1-carboxamide, SULFATE ION, ... (4 entities in total) |
Functional Keywords | ethr, transcription, inhibition |
Biological source | Mycobacterium tuberculosis |
Total number of polymer chains | 1 |
Total formula weight | 24400.25 |
Authors | Tomlinson, C.W.E.,Tatum, N.J.,Pohl, E. (deposition date: 2021-02-09, release date: 2022-02-23, Last modification date: 2024-01-31) |
Primary citation | Tatum, N.J.,Tomlinson, C.W.E.,Frita, R.,Bennett, R.,Baulard, A.R.,Pohl, E.,Kitching, M.O. Systematic exploration of the hydrophobic capacity of the EthR binding site for lead compound optimization To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.26 Å) |
Structure validation
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