7NAA
Crystal structure of Mycobacterium tuberculosis H37Rv PknF kinase domain
Summary for 7NAA
Entry DOI | 10.2210/pdb7naa/pdb |
Descriptor | Non-specific serine/threonine protein kinase, (4-{[4-(1-benzothiophen-2-yl)pyrimidin-2-yl]amino}phenyl)[4-(pyrrolidin-1-yl)piperidin-1-yl]methanone (3 entities in total) |
Functional Keywords | pknf, mtb, transferase, structural genomics, psi-biology, protein structure initiative, structural genomics consortium, sgc, antimicrobial protein |
Biological source | Mycobacterium tuberculosis |
Total number of polymer chains | 4 |
Total formula weight | 123419.64 |
Authors | Oliveira, A.A.,Cabarca, S.,dos Reis, C.V.,Takarada, J.E.,Counago, R.M.,Balan, A.,Structural Genomics Consortium (SGC) (deposition date: 2021-06-21, release date: 2021-08-04, Last modification date: 2023-10-18) |
Primary citation | Cabarca, S.,Frazao de Souza, M.,Albert de Oliveira, A.,Vignoli Muniz, G.S.,Lamy, M.T.,Vinicius Dos Reis, C.,Takarada, J.,Effer, B.,Souza, L.S.,Iriarte de la Torre, L.,Counago, R.,Pinto Oliveira, C.L.,Balan, A. Structure of the Mycobacterium tuberculosis c PknF and conformational changes induced in forkhead-associated regulatory domains. Curr Res Struct Biol, 3:165-178, 2021 Cited by PubMed: 34382010DOI: 10.1016/j.crstbi.2021.07.001 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.75 Å) |
Structure validation
Download full validation report