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7G8V

ARHGEF2 PanDDA analysis group deposition -- ARHGEF2 and RhoA in complex with Z133716556

Summary for 7G8V
Entry DOI10.2210/pdb7g8v/pdb
Group depositionARHGEF2 PanDDA analysis group deposition (G_1002269)
DescriptorTransforming protein RhoA, Rho guanine nucleotide exchange factor 2, N-[(4R)-3,4-dihydro-2H-1-benzopyran-4-yl]methanesulfonamide, ... (6 entities in total)
Functional Keywordssgc - diamond i04-1 fragment screening, pandda, xchemexplorer, cytosolic protein
Biological sourceHomo sapiens (human)
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Total number of polymer chains2
Total formula weight50832.42
Authors
Bradshaw, W.J.,Katis, V.L.,Bountra, C.,von Delft, F.,Brennan, P.E. (deposition date: 2023-06-22, release date: 2023-07-12)
Primary citationBradshaw, W.J.,Katis, V.L.,Bountra, C.,von Delft, F.,Brennan, P.E.
ARHGEF2 PanDDA analysis group deposition
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.451 Å)
Structure validation

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