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7EIK

RD4-BD1 in complex with LT-872-297

Summary for 7EIK
Entry DOI10.2210/pdb7eik/pdb
DescriptorBromodomain-containing protein 4, 1-[2-methyl-5-[6-(4-methylpiperazin-1-yl)-1H-benzimidazol-2-yl]-4-(1-methylpyrazol-4-yl)-1H-pyrrol-3-yl]ethanone (3 entities in total)
Functional Keywordsinhibitor, brd4, bd1, gene regulation
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight15300.69
Authors
Zheng, W.,Kong, B.,Tang, W.,Zhu, J.,Chen, Y. (deposition date: 2021-03-31, release date: 2022-04-06, Last modification date: 2023-11-29)
Primary citationZheng, W.,Kong, B.,Tang, W.,Zhu, J.,Chen, Y.
RD4-BD1 in complex with LT-872-297
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.7 Å)
Structure validation

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