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7EHW

BRD4-BD1 in complex with LT-642-602

Summary for 7EHW
Entry DOI10.2210/pdb7ehw/pdb
DescriptorBromodomain-containing protein 4, 1-[4-ethyl-2-methyl-5-(6-morpholin-4-yl-1H-benzimidazol-2-yl)-1H-pyrrol-3-yl]ethanone (3 entities in total)
Functional Keywordsinhibitor, brd4, bd1, gene regulation
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight15235.62
Authors
Zheng, W.,Kong, B.,Tang, W.,Zhu, J.,Chen, Y. (deposition date: 2021-03-30, release date: 2022-03-30, Last modification date: 2023-11-29)
Primary citationZheng, W.,Kong, B.,Tang, W.,Zhu, J.,Chen, Y.
BRD4-BD1 in complex with LT-642-602
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.65 Å)
Structure validation

246905

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