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7CB7

1.7A resolution structure of SARS-CoV-2 main protease (Mpro) in complex with broad-spectrum coronavirus protease inhibitor GC376

Summary for 7CB7
Entry DOI10.2210/pdb7cb7/pdb
Descriptor3C-like proteinase, SODIUM ION, (1S,2S)-2-({N-[(benzyloxy)carbonyl]-L-leucyl}amino)-1-hydroxy-3-[(3S)-2-oxopyrrolidin-3-yl]propane-1-sulfonic acid, ... (5 entities in total)
Functional Keywordsmain protease, 3c-like proteinase, protein-inhibitor complex, gc376, viral protein
Biological sourceSevere acute respiratory syndrome coronavirus 2 (2019-nCoV)
Total number of polymer chains2
Total formula weight70246.85
Authors
Wang, Y.C.,Yang, C.S.,Hou, M.H.,Tsai, C.L.,Chou, Y.Z.,Chen, Y.,Hung, M.C. (deposition date: 2020-06-10, release date: 2021-05-05, Last modification date: 2023-11-29)
Primary citationWang, Y.C.,Yang, W.H.,Yang, C.S.,Hou, M.H.,Tsai, C.L.,Chou, Y.Z.,Hung, M.C.,Chen, Y.
Structural basis of SARS-CoV-2 main protease inhibition by a broad-spectrum anti-coronaviral drug.
Am J Cancer Res, 10:2535-2545, 2020
Cited by
PubMed: 32905393
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.69 Å)
Structure validation

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