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7BO2

Notum Fragment_130 (4H-thieno[3,2-c]chromene-2-carboxylic acid)

Summary for 7BO2
Entry DOI10.2210/pdb7bo2/pdb
DescriptorPalmitoleoyl-protein carboxylesterase NOTUM, SULFATE ION, 2-acetamido-2-deoxy-beta-D-glucopyranose, ... (7 entities in total)
Functional Keywordsnotum fragment screen, hydrolase
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight45136.68
Authors
Zhao, Y.,Jones, E.Y. (deposition date: 2021-01-23, release date: 2022-03-02, Last modification date: 2024-01-31)
Primary citationZhao, Y.,Jones, E.Y.
Notum Inhibitor
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.21 Å)
Structure validation

221716

PDB entries from 2024-06-26

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