7AR4
Crystal structure of beta-catenin in complex with cyclic peptide inhibitor
This is a non-PDB format compatible entry.
Summary for 7AR4
Entry DOI | 10.2210/pdb7ar4/pdb |
Descriptor | Catenin beta-1, Cadherin-1, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, ... (5 entities in total) |
Functional Keywords | wnt signaling, peptide inhibitor, protein-peptide interaction, signaling protein |
Biological source | Homo sapiens (Human) More |
Total number of polymer chains | 2 |
Total formula weight | 60401.35 |
Authors | Wendt, M.,Pearce, N.M.,Grossmann, T.N.,Hennig, S. (deposition date: 2020-10-23, release date: 2021-04-07, Last modification date: 2024-01-31) |
Primary citation | Wendt, M.,Bellavita, R.,Gerber, A.,Efrem, N.L.,van Ramshorst, T.,Pearce, N.M.,Davey, P.R.J.,Everard, I.,Vazquez-Chantada, M.,Chiarparin, E.,Grieco, P.,Hennig, S.,Grossmann, T.N. Bicyclic beta-Sheet Mimetics that Target the Transcriptional Coactivator beta-Catenin and Inhibit Wnt Signaling. Angew.Chem.Int.Ed.Engl., 60:13937-13944, 2021 Cited by PubMed: 33783110DOI: 10.1002/anie.202102082 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.6 Å) |
Structure validation
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