7QDQ
Crystal Structure of HDM2 in complex with Caylin-1
Summary for 7QDQ
Entry DOI | 10.2210/pdb7qdq/pdb |
Descriptor | E3 ubiquitin-protein ligase Mdm2, CHLORIDE ION, SODIUM ION, ... (7 entities in total) |
Functional Keywords | nmr molecular replacement, complex structure, drug design, nmr spectroscopy, structure elucidation, ligase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 11825.68 |
Authors | Finke, A.D.,Walti, M.A.,Marsh, M.E.,Orts, J. (deposition date: 2021-11-29, release date: 2022-10-05, Last modification date: 2024-02-07) |
Primary citation | Mertens, V.,Abi Saad, M.J.,Coudevylle, N.,Walti, M.A.,Finke, A.,Marsh, M.,Orts, J. Elucidation of a nutlin-derivative-HDM2 complex structure at the interaction site by NMR molecular replacement: A straightforward derivation J Magn Reson Open, 10-11:100032-, 2022 Cited by DOI: 10.1016/j.jmro.2022.100032PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.26 Å) |
Structure validation
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