6YK1
Crystal structure of mouse pyridoxal kinase in complex with ATP-gamma-S and artesunate
Summary for 6YK1
Entry DOI | 10.2210/pdb6yk1/pdb |
Descriptor | Pyridoxal kinase, GLYCEROL, TETRAETHYLENE GLYCOL, ... (7 entities in total) |
Functional Keywords | pdxk, plp, pl, vitamin b6, enzyme, artemisinin, artesunate, transferase |
Biological source | Mus musculus (Mouse) |
Total number of polymer chains | 4 |
Total formula weight | 145687.39 |
Authors | Kasaragod, V.B.,Schindelin, H. (deposition date: 2020-04-05, release date: 2021-04-14, Last modification date: 2024-01-24) |
Primary citation | Kasaragod, V.B.,Pacios-Michelena, A.,Schaefer, N.,Zheng, F.,Bader, N.,Alzheimer, C.,Villmann, C.,Schindelin, H. Pyridoxal kinase inhibition by artemisinins down-regulates inhibitory neurotransmission. Proc.Natl.Acad.Sci.USA, 117:33235-33245, 2020 Cited by PubMed: 33318193DOI: 10.1073/pnas.2008695117 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.4 Å) |
Structure validation
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