6YH1
tRNA-guanine Transglycosylase (TGT) labeled with 5-fluorotryptophan in co-crystallized complex with 6-amino-2-(methylamino)-4-(4-(trifluoromethyl)phenethyl)-3,7-dihydro-8H-imidazo[4,5-g]quinazolin-8-one
Summary for 6YH1
Entry DOI | 10.2210/pdb6yh1/pdb |
Related | 6YGS |
Descriptor | Queuine tRNA-ribosyltransferase, ZINC ION, 6-amino-2-(methylamino)-4-(4-(trifluoromethyl)phenethyl)-3,7-dihydro-8H-imidazo[4,5-g]quinazolin-8-one, ... (4 entities in total) |
Functional Keywords | transferase, tgt, trna-guanine transglycosylase, guanine insertion enzyme, homodimer, 19f nmr |
Biological source | Zymomonas mobilis subsp. mobilis ZM4 = ATCC 31821 |
Total number of polymer chains | 1 |
Total formula weight | 43609.57 |
Authors | Nguyen, A.,Heine, A.,Klebe, G. (deposition date: 2020-03-28, release date: 2020-04-08, Last modification date: 2024-01-24) |
Primary citation | Nguyen, A.,Heine, A.,Klebe, G. Co-crystallization, nanoESI-MS and 19F NMR reveal dimer disturbing inhibitors and conformational changes at dimer contacts To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.55 Å) |
Structure validation
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