6SQM

Crystal structure of CREBBP bromodomain complexed with LA36

Summary for 6SQM

• Entry DOI: 10.2210/pdb6sqm/pdb
• Descriptor: CREB-binding protein, ~{N}-[3-acetamido-5-[(3-methylcinnolin-5-yl)carbamoyl]phenyl]furan-2-carboxamide, 1,2-ETHANEDIOL, ... (4 entities in total)
• Functional Keywords: inhibitor, complex, crebbp, bromodomain, transferase
• Biological source: Homo sapiens (Human)
• Total number of polymer chains: 3
• Total formula weight: 44144.53

Authors

Bedi, R.K.,Laul, E.,Nevado, C.,Caflisch, A. (deposition date: 2019-09-04, release date: 2020-09-30, Last modification date: 2024-01-24)

• Primary citation: Bedi, R.K.,Laul, E.,Nevado, C.,Caflisch, A.; Crystal structure of CREBBP bromodomain complexed with LA36; To Be Published,

Experimental method

X-RAY DIFFRACTION (1.8 Å)