6RCH
Crystal structure of Casein kinase I isoform delta (CK1 delta) complexed with SR4133 inhibitor
Summary for 6RCH
Entry DOI | 10.2210/pdb6rch/pdb |
Descriptor | Casein kinase I isoform delta, SULFATE ION, 1,2-ETHANEDIOL, ... (6 entities in total) |
Functional Keywords | ck1 delta, ck1d, kinase inhibitor, structural genomics, structural genomics consortium, sgc, transferase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 2 |
Total formula weight | 70452.95 |
Authors | Chaikuad, A.,Arrowsmith, C.H.,Edwards, A.M.,Bountra, C.,Roush, W.R.,Knapp, S.,Structural Genomics Consortium (SGC) (deposition date: 2019-04-11, release date: 2020-03-25, Last modification date: 2024-01-24) |
Primary citation | Chaikuad, A.,Arrowsmith, C.H.,Edwards, A.M.,Bountra, C.,Roush, W.R.,Knapp, S.,Structural Genomics Consortium (SGC) Crystal structure of Casein kinase I isoform delta (CK1 delta) complexed with SR4133 inhibitor To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.45 Å) |
Structure validation
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