6RCG
Crystal structure of Casein kinase 1 delta (CK1 delta) complexed with SR3029 inhibitor
Summary for 6RCG
Entry DOI | 10.2210/pdb6rcg/pdb |
Descriptor | Casein kinase I isoform delta, 1,2-ETHANEDIOL, ~{N}-[[6,7-bis(fluoranyl)-1~{H}-benzimidazol-2-yl]methyl]-9-(3-fluorophenyl)-2-morpholin-4-yl-purin-6-amine, ... (4 entities in total) |
Functional Keywords | csnk1d, ck1 delta, ck1d, kinase inhibitor, structural genomics, structural genomics consortium, sgc, transferase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 35029.39 |
Authors | Chaikuad, A.,Arrowsmith, C.H.,Edwards, A.M.,Bountra, C.,Roush, W.R.,Knapp, S.,Structural Genomics Consortium (SGC) (deposition date: 2019-04-11, release date: 2020-03-25, Last modification date: 2024-01-24) |
Primary citation | Chaikuad, A.,Arrowsmith, C.H.,Edwards, A.M.,Bountra, C.,Roush, W.R.,Knapp, S.,Structural Genomics Consortium (SGC) Crystal structure of Casein kinase 1 delta (CK1 delta) complexed with SR3029 inhibitor To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.4 Å) |
Structure validation
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