6QDX
Structure of E.coli RlmJ in complex with a bisubstrate analogue (BA4)
Summary for 6QDX
Entry DOI | 10.2210/pdb6qdx/pdb |
Descriptor | Ribosomal RNA large subunit methyltransferase J, (2~{S})-4-[[(2~{S},3~{S},4~{R},5~{R})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl-[3-[[9-[(2~{S},3~{R},4~{S},5~{S})-5-(hydroxymethyl)-3,4-bis(oxidanyl)oxolan-2-yl]purin-6-yl]amino]propyl]amino]-2-azanyl-butanoic acid (3 entities in total) |
Functional Keywords | rna mtases, methyltransferase, m6a, transition state analogue, inhibitor, rna binding, trmk, rlmj, m1a, structure., transferase |
Biological source | Escherichia coli |
Total number of polymer chains | 4 |
Total formula weight | 131786.48 |
Authors | Oerum, S.,Catala, M.,Atdjian, C.,Brachet, F.,Ponchon, L.,Barraud, P.,Iannazzo, L.,Droogmans, L.,Braud, E.,Etheve-Quelquejeu, M.,Tisne, C. (deposition date: 2019-01-03, release date: 2019-03-27, Last modification date: 2024-01-24) |
Primary citation | Oerum, S.,Catala, M.,Atdjian, C.,Brachet, F.,Ponchon, L.,Barraud, P.,Iannazzo, L.,Droogmans, L.,Braud, E.,Etheve-Quelquejeu, M.,Tisne, C. Bisubstrate analogues as structural tools to investigate m6A methyltransferase active sites. Rna Biol., 16:798-808, 2019 Cited by PubMed: 30879411DOI: 10.1080/15476286.2019.1589360 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.1 Å) |
Structure validation
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