6Q7V
Crystal structure of PqsR (MvfR) ligand-binding domain in complex with compound 11
Summary for 6Q7V
Entry DOI | 10.2210/pdb6q7v/pdb |
Descriptor | Transcriptional regulator MvfR, ~{N}4-[(4-fluorophenyl)methyl]-6-(trifluoromethyl)pyridine-2,4-diamine (3 entities in total) |
Functional Keywords | quorum sensing, lysr-type transcriptional regulator, pseudomonas quinolone signaling system, lttr, dna binding protein |
Biological source | Pseudomonas aeruginosa PAO1 |
Total number of polymer chains | 2 |
Total formula weight | 51970.62 |
Authors | Witzgall, F.,Blankenfeldt, W. (deposition date: 2018-12-13, release date: 2019-11-20, Last modification date: 2024-01-24) |
Primary citation | Zender, M.,Witzgall, F.,Kiefer, A.,Kirsch, B.,Maurer, C.K.,Kany, A.M.,Xu, N.,Schmelz, S.,Borger, C.,Blankenfeldt, W.,Empting, M. Flexible Fragment Growing Boosts Potency of Quorum-Sensing Inhibitors against Pseudomonas aeruginosa Virulence. Chemmedchem, 15:188-194, 2020 Cited by PubMed: 31709767DOI: 10.1002/cmdc.201900621 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.56 Å) |
Structure validation
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